SCHEMBL27675176

SCHEMBL27675176

C=CC(N1CCOCC1)S(=O)(=O)c1cccc(N)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.42
ALDH1A1 P00352 2/20 0.42
HSD17B10 Q99714 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
PKM P14618 6/20 0.41
LMNA P02545 1/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA4 P22748 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
PKLR P30613 1/20 0.38
HPGD P15428 1/20 0.35
F2 P00734 1/20 0.35
PRSS1 P07477 1/20 0.35
PRSS2 P07478 1/20 0.35
PRSS3 P35030 1/20 0.35
POLB P06746 1/20 0.34
RECQL P46063 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27693671 0.87 ALDH1A1 (0.44) TSHRALDH1A1HSD17B10TDP1PKM
SCHEMBL27669965 0.85 ADRA2C (0.42) TSHRALDH1A1HSD17B10TDP1PKM
SCHEMBL27743079 0.85 PKM (0.41) ALDH1A1HSD17B10PKMLMNAPKLR
SCHEMBL27693489 0.84 POLB (0.36) TSHRALDH1A1TDP1PKMLMNA
SCHEMBL27735019 0.84 PKM (0.45) TSHRALDH1A1HSD17B10PKMLMNA
SCHEMBL27755443 0.82 ALDH1A1 (0.40) TSHRALDH1A1HSD17B10TDP1PKM
SCHEMBL27754807 0.80 TSHR (0.42) TSHRALDH1A1HSD17B10PKMLMNA
SCHEMBL27745075 0.80 CA1 (0.43) TSHRALDH1A1LMNACA12CA1
SCHEMBL27835248 0.78 LMNA (0.37) ALDH1A1LMNAPOLB
Hydrochloric Acid SCHEMBL27739197 0.77 CA2 (0.40) ALDH1A1LMNACA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101006076-B Modulators of ATP-binding cassette transporters VERTEX PHARMA 2010-09-29 CN disclosed
CN-100528876-C Pyrrazolo-pyrimidine derivatives HOFFMANN LA ROCHE (CH) 2009-08-19 CN disclosed
CN-101006076-A Modulators of ATP-binding cassette transporters VERTEX PHARMA (US) 2007-07-25 CN disclosed
CN-1964973-A Pyrrazolo-pyrimidine derivatives HOFFMANN LA ROCHE (CH) 2007-05-16 CN disclosed