SCHEMBL27675217

SCHEMBL27675217

CCOC(=O)c1ccccc1-c1ccc([N+](=O)[O-])c([N+](=O)[O-])c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.50
SMN1; SMN2 Q16637 3/20 0.50
LMNA P02545 2/20 0.50
POLB P06746 2/20 0.50
GALR2 O43603 1/20 0.50
MITF O75030 1/20 0.50
HSP90AA1 P07900 1/20 0.50
HPGD P15428 1/20 0.50
XBP1 P17861 1/20 0.50
CCR6 P51684 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
TSHR P16473 1/20 0.50
MAPT P10636 5/20 0.49
GAA P10253 1/20 0.49
HTT P42858 1/20 0.48
ERN1 O75460 1/20 0.46
HSD17B10 Q99714 1/20 0.44
CACNA1D Q01668 2/20 0.44
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31325723 0.88 ERN1 (0.54) ALDH1A1SMN1; SMN2LMNATSHRMAPT
SCHEMBL27636819 0.85 SLC6A3 (0.59) ALDH1A1SMN1; SMN2LMNAMAPTHTT
SCHEMBL7640668 0.83 MAPT (0.57) SMN1; SMN2POLBTSHRMAPTGAA
SCHEMBL27585698 0.79 CASP6 (0.51) ALDH1A1SMN1; SMN2TSHR
SCHEMBL15847247 0.79 ALDH1A1 (0.51) ALDH1A1SMN1; SMN2LMNAPOLBGALR2
SCHEMBL1523174 0.79 ALDH1A1 (0.67) ALDH1A1SMN1; SMN2LMNAPOLBGALR2
SCHEMBL27647715 0.78 BCAT2 (0.53) ALDH1A1LMNAPOLBMAPTERN1
SCHEMBL27845352 0.78 CTSD (0.43) ALDH1A1POLBTSHRMAPTHSD17B10
SCHEMBL27675256 0.78 MAPT (0.55) ALDH1A1SMN1; SMN2LMNAPOLBGALR2
SCHEMBL7984053 0.78 ALDH1A1 (0.50) ALDH1A1SMN1; SMN2LMNAPOLBGALR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102652128-A 4-Oxo-1H-quinoline-3-carboxamides as modulators of ATP-binding cassette transporters VERTEX PHARMA 2012-08-29 CN disclosed
CN-101006076-B Modulators of ATP-binding cassette transporters VERTEX PHARMA 2010-09-29 CN disclosed
CN-101006076-A Modulators of ATP-binding cassette transporters VERTEX PHARMA (US) 2007-07-25 CN disclosed