SCHEMBL27675673

SCHEMBL27675673

CCOc1cc[c]cc1N(C)C

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.33
NQO1 P15559 1/20 0.32
KDM4E B2RXH2 4/20 0.32
L3MBTL1 Q9Y468 3/20 0.32
KMT2A Q03164 2/20 0.32
MAPT P10636 2/20 0.32
HPGD P15428 2/20 0.32
MEN1 O00255 1/20 0.32
POLB P06746 1/20 0.32
MAPK1 P28482 1/20 0.32
HSD17B10 Q99714 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.31
PDE4A P27815 1/20 0.30
PDE4B Q07343 1/20 0.30
PDE4C Q08493 1/20 0.30
PDE4D Q08499 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
GLA P06280 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27650969 0.86 ALDH1A1 (0.34) ALDH1A1KDM4EKMT2AMAPTMEN1
SCHEMBL5664732 0.85 ALDH1A1 (0.33) ALDH1A1NQO1KDM4EL3MBTL1KMT2A
SCHEMBL27813748 0.84 CCR5 (0.33) ALDH1A1NQO1KDM4EL3MBTL1KMT2A
SCHEMBL8106329 0.82 THRA (0.39) ALDH1A1KMT2AMAPTHPGDMEN1
SCHEMBL7356480 0.81 CCR5 (0.31)
SCHEMBL6584974 0.79 APP (0.40)
SCHEMBL127280 0.78 ALDH1A1 (0.39) ALDH1A1NQO1KDM4EL3MBTL1KMT2A
SCHEMBL1231501 0.76 ALDH1A1 (0.38) ALDH1A1NQO1KDM4EL3MBTL1KMT2A
SCHEMBL596846 0.73 L3MBTL1 (0.39) ALDH1A1NQO1KDM4EL3MBTL1KMT2A
SCHEMBL3043536 0.73 ALDH1A1 (0.40) ALDH1A1NQO1KDM4EL3MBTL1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101912400-B 5-amino-2,4,7-trioxo-3,4,7,8-tetrahydro-2h-pyrido[2,3-d] pyrimidine derivatives and related compounds for the treatment of cancer JAPAN TOBACCO INC 2013-06-26 CN disclosed
CN-1809570-B [1,2,4] triazolo [1,5-a ] pyrimidin-2-ylurea derivatives and uses thereof NIPPON KAYAKU KK 2011-06-22 CN disclosed
CN-101912400-A The 5-amino-2,4 that is used for the treatment of cancer, 7-trioxy--3,4,7,8-tetrahydrochysene-2H-pyrido [2,3-d] pyrimidine derivatives and related compound JAPAN TOBACCO INC 2010-12-15 CN disclosed
CN-101006086-B 5-amino-2, 4, 7-trioxo-3, 4,7, 8-tetrahydro-2H-pyrido [2,3-d ] pyrimidine derivatives and related compounds for the treatment of cancer JAPAN TOBACCO INC 2010-09-29 CN disclosed
CN-101006086-A 5-amino-2, 4, 7-trioxo-3, 4,7, 8-tetrahydro-2H-pyrido [2, 3-d ] pyrimidine derivatives and related compounds for the treatment of cancer JAPAN TOBACCO INC (JP) 2007-07-25 CN disclosed