SCHEMBL28024448

SCHEMBL28024448

Cc1cc(N)ccc1C1CCN(OC(=O)C(C)(C)C)CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 1/20 0.36
NR1H2 P55055 1/20 0.36
HTR1D P28221 1/20 0.34
HTR1B P28222 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
SLC9A1 P19634 1/20 0.34
CYP2C19 P33261 1/20 0.34
KCNH2 Q12809 1/20 0.34
RAD52 P43351 1/20 0.34
DRD4 P21917 1/20 0.34
PROKR1 Q8TCW9 2/20 0.34
FAAH O00519 1/20 0.33
CRBN Q96SW2 1/20 0.33
MAPT P10636 2/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
THRB P10828 1/20 0.33
NR4A1 P22736 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28024911 0.86 GPR119 (0.40) OPRL1NR1H2HTR1DHTR1BCYP3A4
SCHEMBL28839896 0.85 NR1H2 (0.34) NR1H2HTR1DHTR1BCYP3A4CYP2C9
SCHEMBL27948292 0.84 SLC9A1 (0.48) CYP3A4CYP2C9SLC9A1CYP2C19KCNH2
SCHEMBL30021635 0.81 MAPT (0.51) NR1H2MAPTMEN1ALDH1A1THRB
SCHEMBL1159547 0.81 MAPT (0.51) NR1H2MAPTMEN1ALDH1A1THRB
SCHEMBL27682015 0.81 RIPK1 (0.39) CRBN
SCHEMBL27318172 0.80 SLC18A3 (0.44) CYP3A4CYP2C9CRBN
SCHEMBL28053666 0.79 HTR1D (0.63) HTR1DHTR1BCYP3A4CYP2C9MAPT
SCHEMBL27944975 0.78 MAPT (0.52) NR1H2RAD52MAPTMEN1ALDH1A1
SCHEMBL27915293 0.78 TRPC6 (0.36) TRPC6TRPV1SSTR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105829315-B Pyrimidopyrimidinones useful as Wee-1 kinase inhibitors 阿尔麦克探索有限公司 2019-03-08 CN disclosed
CN-105829315-A Pyrimidopyrimidinones useful as Wee-1 kinase inhibitors 阿尔麦克探索有限公司 2016-08-03 CN disclosed
CN-104837835-A VEGFR3 inhibitors CANCER THERAPEUTICS CRC PTY LTD 2015-08-12 CN disclosed