SCHEMBL2768765

SCHEMBL2768765

COc1ccc(N2CCN(CCC3CCCCC3)CC2)cc1F

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 2/20 0.47
HTR2C P28335 2/20 0.46
DRD2 P14416 5/20 0.46
DRD3 P35462 5/20 0.46
CTSL P07711 1/20 0.44
CTSS P25774 1/20 0.44
CTSK P43235 1/20 0.44
HTR2A P28223 1/20 0.42
HTR7 P34969 1/20 0.42
KDM4E B2RXH2 1/20 0.42
ACHE P22303 1/20 0.41
HTR4 Q13639 1/20 0.41
HTR1A P08908 1/20 0.41
DRD4 P21917 1/20 0.41
HTR2B P41595 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2766456 0.82 FFAR4 (0.48) DRD2DRD3HTR7ACHEHTR4
SCHEMBL2768705 0.81 DRD2 (0.48) DRD2DRD3
SCHEMBL23102236 0.78 KDM4E (0.50) DRD2DRD3HTR7KDM4EACHE
SCHEMBL17241036 0.77 ALDH1A1 (0.54) HTR2CKDM4E
SCHEMBL2767452 0.76 SLC6A2 (0.46) CHRM4DRD2DRD3CTSLCTSS
SCHEMBL14922721 0.76 SIRT6 (0.55) DRD2DRD3HTR2AKDM4EHTR1A
SCHEMBL2768860 0.76 ADRA1D (0.61) DRD2HTR1A
SCHEMBL2766482 0.75 FFAR4 (0.47) HTR2CDRD2DRD3HTR2AHTR7
SCHEMBL2768242 0.75 SLC6A2 (0.47) CHRM4DRD2DRD3
SCHEMBL2766690 0.75 DRD2 (0.42) HTR2CDRD2DRD3HTR2AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1627871-B1 CYCLIC AMINOPHENYL SULFAMATE DERIVATIVE ASKA PHARM CO LTD (JP) 2010-04-14 EP disclosed
US-7449466-B2 Cyclic aminophenyl sulfamate derivative ASKA PHARMACEUTICAL CO., LTD. (JP) 2008-11-11 US disclosed
US-20060189625-A1 Cyclic aminophenyl sulfamate derivative ASKA PHARMACEUTICAL CO., LTD. (JP) 2006-08-24 US disclosed
EP-1627871-A1 CYCLIC AMINOPHENYL SULFAMATE DERIVATIVE Teikoku Hormone Mfg. Co., Ltd. (JP) 2006-02-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060189625-A1 Cyclic aminophenyl sulfamate derivative SHBG, STS, ARSA CHRM4 1818/4885HTR2C 1544/4885DRD2 3225/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.