SCHEMBL27694580

SCHEMBL27694580

C=CC(c1ccc(S(C)(=O)=O)cc1)S(=O)(=O)CCC1(O)CCN(C(=O)O)CC1

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
S1PR2 O95136 5/20 0.35
CCR5 P51681 6/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
OPRM1 P35372 2/20 0.32
OPRD1 P41143 2/20 0.32
OPRK1 P41145 2/20 0.32
OPRL1 P41146 2/20 0.32
LMNA P02545 1/20 0.32
GPR119 Q8TDV5 1/20 0.32
DPP4 P27487 1/20 0.32
DPP7 Q9UHL4 1/20 0.32
TGM2 P21980 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27694589 0.90 CCR5 (0.33) CCR5LMNAGPR119DPP4DPP7
SCHEMBL27694627 0.89 CCR5 (0.33) S1PR2CCR5LMNAGPR119DPP4
SCHEMBL27676117 0.83 TGM2 (0.31) TGM2
SCHEMBL4977808 0.80 KMT2A (0.41) S1PR2ALDH1A1KMT2AL3MBTL1LMNA
SCHEMBL27694579 0.74 MAOB (0.36) S1PR2ALDH1A1KMT2AL3MBTL1LMNA
SCHEMBL28763206 0.73 OPRD1 (0.32) OPRD1
SCHEMBL27676119 0.72 PTGS1 (0.32)
SCHEMBL27694590 0.71 PTGS2 (0.34) OPRD1
SCHEMBL27694630 0.69 CTSK (0.31)
SCHEMBL4978743 0.68 LMNA (0.38) CCR5KMT2ALMNAGPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101006057-A Novel piperidine/8-azabicyclo [3.2.1] octan derivatives as moduilators of chemokine receptor CCR5 ASTRAZENECA AB (SE) 2007-07-25 CN disclosed