SCHEMBL27706331

SCHEMBL27706331

O=C(NNc1cccnc1)OCc1ccccc1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 2/20 0.60
P2RX7 Q99572 1/20 0.59
KMT2A Q03164 3/20 0.57
LMNA P02545 2/20 0.57
POLB P06746 1/20 0.57
TDP1 Q9NUW8 1/20 0.57
MEN1 O00255 2/20 0.54
SGMS2 Q8NHU3 1/20 0.53
CHRNA7 P36544 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
GRIN2B Q13224 1/20 0.52
GAA P10253 1/20 0.51
ALDH1A1 P00352 1/20 0.50
MAPT P10636 1/20 0.50
HTT P42858 1/20 0.50
NPC1 O15118 1/20 0.49
PKM P14618 1/20 0.49
RAB9A P51151 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL968903 0.87 POLB (0.71) NAMPTKMT2ALMNAPOLBTDP1
SCHEMBL4908338 0.85 GAA (0.69) P2RX7KMT2ALMNAPOLBTDP1
SCHEMBL11563747 0.81 NAMPT (0.77) NAMPTKMT2ALMNAPOLBTDP1
SCHEMBL27532876 0.79 KDM4E (0.51) NAMPTP2RX7KMT2ALMNAPOLB
SCHEMBL7742679 0.78 NAMPT (0.68) NAMPTKMT2ALMNATDP1CYP3A4
SCHEMBL1665313 0.78 POLB (0.67) NAMPTKMT2ALMNAPOLBMEN1
SCHEMBL5348225 0.78 ALDH1A1 (0.60) NAMPTKMT2ALMNAPOLBTDP1
SCHEMBL27775337 0.77 P2RX7 (0.66) NAMPTP2RX7KMT2ALMNAPOLB
SCHEMBL9130883 0.76 NPC1 (0.58) NAMPTP2RX7LMNAGAAALDH1A1
SCHEMBL5347283 0.76 KMT2A (0.63) NAMPTKMT2ALMNAPOLBTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110511209-A It can be used as the indole carboxamides compound of kinase inhibitor BRISTOL MYERS SQUIBB CO 2019-11-29 CN disclosed
CN-107108583-A Indole carboxamide compounds useful as kinase inhibitors 百时美施贵宝公司 2017-08-29 CN disclosed
CN-103073460-B Be applicable to treat the aromatic substance that the arylsulfonyl ylmethyl of the disease responded for the adjustment of dopamine D 3 receptor or aryl sulfonic acid amides replace AbbVie Deutschland GmbH & Co. KG (DE) 2015-09-09 CN disclosed
CN-102112447-B HIV integrase inhibitors from pyridoxine AMBRILIA BIOPHARMA INC 2013-06-26 CN disclosed
CN-103073460-A Arylsulfonylmethyl or arylsulfonamide substituted aromatic compounds suitable for treating disorders that respond to modulation of the dopamine D3 receptor ABBOTT GMBH & CO KG 2013-05-01 CN disclosed
CN-101068801-B Arylsulfonylmethyl or arylsulfonamide substituted aromatic compounds suitable for the treatment of disorders which respond to modulation of the dopamine D3 receptor ABBOTT GMBH & CO KG 2012-11-14 CN disclosed
CN-102112447-A HIV integrase inhibitors from pyridoxine AMBRILIA BIOPHARMA INC 2011-06-29 CN disclosed
CN-101678022-A 5-cyano-4- (pyrrolo [2,3b ] pyridin-3-yl) pyrimidine derivatives useful as protein kinase inhibitors VERTEX PHARMA 2010-03-24 CN disclosed
CN-101068801-A Arylsulfonylmethyl or arylsulfonamide substituted aromatic compounds suitable for the treatment of disorders which respond to modulation of the dopamine D3 receptor ABBOTT GMBH & CO KG (DE) 2007-11-07 CN disclosed