SCHEMBL9130883

SCHEMBL9130883

O=C(O)NNc1cccnc1

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.58
RAB9A P51151 4/20 0.58
PKM P14618 1/20 0.58
P2RX7 Q99572 1/20 0.55
NAMPT P43490 6/20 0.54
ALDH1A1 P00352 3/20 0.51
LMNA P02545 2/20 0.51
HIF1A Q16665 1/20 0.51
KDM4E B2RXH2 1/20 0.51
HTT P42858 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
GAA P10253 1/20 0.49
TP53 P04637 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19322921 0.83 CYP3A4 (0.60) NPC1RAB9APKMP2RX7NAMPT
SCHEMBL27532876 0.80 KDM4E (0.51) NPC1RAB9APKMP2RX7NAMPT
SCHEMBL29136551 0.80 P2RX7 (0.51) NPC1RAB9APKMP2RX7NAMPT
SCHEMBL967245 0.80 RAB9A (0.72) NPC1RAB9APKMNAMPTALDH1A1
SCHEMBL11213715 0.80 RAB9A (0.72) NPC1RAB9APKMNAMPTALDH1A1
SCHEMBL19318495 0.79 TSHR (0.58) NPC1RAB9APKMP2RX7NAMPT
SCHEMBL4718965 0.77 ALDH1A1 (0.57) NPC1RAB9APKMNAMPTALDH1A1
SCHEMBL3724442 0.77 ALOX5 (0.67) ALDH1A1LMNAKDM4EGAATP53
SCHEMBL19519086 0.76 ALDH1A1 (0.51) NPC1RAB9APKMP2RX7NAMPT
SCHEMBL27706331 0.76 NAMPT (0.60) NPC1RAB9APKMP2RX7NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102656159-A Cgrp receptor antagonists BRISTOL MYERS SQUIBB CO 2012-09-05 CN claimed
US-5411967-A Antiinflammatory, immunosuppressant, antitumor AMERICAN HOME PRODUCTS CORPORATION (US) 1995-05-02 US claimed
CN-106517049-B 360 ° of large parts turnover devices of one kind and its working method 江苏建筑职业技术学院 2018-07-20 CN disclosed
CN-107108583-A Indole carboxamide compounds useful as kinase inhibitors 百时美施贵宝公司 2017-08-29 CN disclosed
CN-102656159-A Cgrp receptor antagonists BRISTOL MYERS SQUIBB CO 2012-09-05 CN disclosed
CN-101855222-A Imidazol (1,2-A)pyridines and related compounds with activity at cannabinoid CB2 receptors GE HEALTHCARE LTD 2010-10-06 CN disclosed
CN-101730691-A Nitrogen-containing aromatic six-membered ring derivatives and drugs containing the same ASUBIO PHARMA CO LTD 2010-06-09 CN disclosed
CN-100579979-C 7-phenylpyrazolopyridine compounds EISAI R&D MAN CO LTD 2010-01-13 CN disclosed
CN-101081850-A 7-phenylpyrazolopyridine compounds EISAI CO LTD (JP) 2007-12-05 CN disclosed
CN-101081853-A 4- (hydroxymethyl) -2, 6-dimethoxyphenylboronic acid compound EISAI CO LTD (JP) 2007-12-05 CN disclosed
CN-1705665-A 7-phenylpyrazolopyridine compounds EISAI CO LTD (JP) 2005-12-07 CN disclosed
US-5411967-A Antiinflammatory, immunosuppressant, antitumor AMERICAN HOME PRODUCTS CORPORATION (US) 1995-05-02 US disclosed