SCHEMBL27736992

SCHEMBL27736992

CN1CCN(C(C=O)CCl)CC1

nearest known ligand 0.31

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.31
CHRM4 P08173 1/20 0.31
CHRM5 P08912 1/20 0.31
ADRA2A P08913 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
CYP2D6 P10635 1/20 0.31
CHRM1 P11229 1/20 0.31
CHRM3 P20309 1/20 0.31
DRD1 P21728 1/20 0.31
ADRA1D P25100 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
HRH1 P35367 1/20 0.31
OPRM1 P35372 1/20 0.31
DRD3 P35462 1/20 0.31
HTR2B P41595 1/20 0.31
SLC6A3 Q01959 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23668191 0.81 HTR1A (0.31) CHRM2CHRM4CHRM5ADRA2AADORA3
SCHEMBL27896230 0.79 NCF1 (0.31) CHRM2CHRM4CHRM5ADRA2AADORA3
SCHEMBL27736373 0.77 ALDH1A1 (0.37) CHRM2CHRM1DRD3
SCHEMBL18390314 0.76 MC4R (0.32)
SCHEMBL8211301 0.76
SCHEMBL27587337 0.75 MAPT (0.36)
SCHEMBL7036171 0.75 MAPT (0.33) CHRM2CHRM4CHRM5ADRA2AADORA3
SCHEMBL27757050 0.75 SIGMAR1 (0.31)
SCHEMBL27737501 0.72 SIGMAR1 (0.35) CHRM2CHRM1
SCHEMBL4629370 0.71 CHRM2 (0.33) CHRM2CHRM4CHRM5ADRA2AADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101367794-B Preparation method for quinazoline derivants and medical uses thereof SHANGHAI HENGRUI PHARM CO LTD 2013-07-10 CN disclosed
CN-102295636-A Indol-3-y-carbonyl-piperidin and piperazin-derivatives 2011-12-28 CN disclosed
CN-101367794-A Preparation method for quinazoline derivants and medical uses thereof SHANGHAI HENGRUI PHARM CO LTD (CN) 2009-02-18 CN disclosed
CN-101277945-A Indol-3-yl-carbonyl-piperidine and piperazine derivatives HOFFMANN LA ROCHE (CH) 2008-10-01 CN disclosed