SCHEMBL27744709

SCHEMBL27744709

O=C(Nc1cccnc1)c1ccccc1Nc1ccccc1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.67
ALDH1A1 P00352 4/20 0.67
MEN1 O00255 3/20 0.67
KMT2A Q03164 3/20 0.67
KDM4E B2RXH2 2/20 0.67
HPGD P15428 1/20 0.67
CYP11B2 P19099 2/20 0.65
NAMPT P43490 3/20 0.63
HSD17B10 Q99714 2/20 0.61
MAPK1 P28482 1/20 0.61
SIRT2 Q8IXJ6 1/20 0.61
PKM P14618 2/20 0.60
TDP1 Q9NUW8 1/20 0.60
LMNA P02545 3/20 0.59
HTT P42858 1/20 0.59
L3MBTL1 Q9Y468 1/20 0.59
NPC1 O15118 2/20 0.58
RAB9A P51151 2/20 0.58
SGMS2 Q8NHU3 1/20 0.57
GAA P10253 2/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5698795 0.87 PKM (0.77) TSHRALDH1A1MEN1KMT2AKDM4E
SCHEMBL24074161 0.84 TSHR (0.74) TSHRALDH1A1MEN1KMT2AKDM4E
SCHEMBL18132518 0.83 ALDH1A1 (0.72) TSHRALDH1A1MEN1KMT2AKDM4E
SCHEMBL28741286 0.83 FABP4 (0.65) TSHRALDH1A1MEN1KMT2AKDM4E
SCHEMBL14396861 0.83 BRAF (0.58) TSHRALDH1A1MEN1KMT2AKDM4E
SCHEMBL24074163 0.82 TSHR (0.70) TSHRALDH1A1MEN1KMT2AKDM4E
SCHEMBL28687927 0.81 CYP11B2 (0.67) TSHRALDH1A1MEN1KMT2AKDM4E
SCHEMBL30322828 0.80 MEN1 (1.00) TSHRALDH1A1MEN1KMT2AKDM4E
SCHEMBL5311227 0.80 MEN1 (1.00) TSHRALDH1A1MEN1KMT2AKDM4E
SCHEMBL6774617 0.79 CHRNB2 (0.71) ALDH1A1MEN1KMT2AKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101321529-B Diaryl aether derivant as antineoplastic agent OTSUKA PHARMA CO LTD 2012-09-05 CN disclosed
CN-101321529-A Diaryl aether derivant as antineoplastic agent OTSUKA PHARMA CO LTD (JP) 2008-12-10 CN disclosed