SCHEMBL27747745

SCHEMBL27747745

CN1CCCC1CCn1ccc2cc(N)ccc21.Cc1c(C(=O)O)cccc1C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 11/20 0.49
NOS1 P29475 11/20 0.49
NOS2 P35228 8/20 0.49
HTR6 P50406 4/20 0.43
CHRNB2 P17787 1/20 0.42
CHRNA4 P43681 1/20 0.42
CHRM3 P20309 1/20 0.42
NTSR1 P30989 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12367568 0.86 NOS3 (0.56) NOS3NOS1NOS2HTR6CHRNB2
SCHEMBL27768895 0.85 CHRNB2 (0.46) NOS3NOS1NOS2HTR6CHRNB2
SCHEMBL27894537 0.83 NTSR1 (0.46) NOS3NOS1NOS2HTR6NTSR1
SCHEMBL2263565 0.82 NOS3 (0.56) NOS3NOS1NOS2HTR6
SCHEMBL1122077 0.77 NOS3 (0.57) NOS3NOS1NOS2HTR6CHRNB2
SCHEMBL2261758 0.76 HTR6 (0.67) NOS3NOS1NOS2HTR6CHRNB2
SCHEMBL2261753 0.76 HTR6 (0.67) NOS3NOS1NOS2HTR6CHRNB2
SCHEMBL2266154 0.73 NOS3 (0.56) NOS3NOS1NOS2HTR6
SCHEMBL8530808 0.72 HTR6 (0.77) NOS3NOS1NOS2HTR6
SCHEMBL2265023 0.72 ADRA2A (0.46) NOS3NOS1NOS2HTR6CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101466709-B 1,5 and 3, 6-substituted indole compounds having NOS inhibitory activity NEURAXON INC 2013-03-20 CN disclosed
CN-101466709-A 1, 5 and 3, 6-substituted indole compounds having NOS inhibitory activity NEURAXON INC (CA) 2009-06-24 CN disclosed