SCHEMBL2776754

SCHEMBL2776754

CN(C)CCC1CCc2cc([N+](=O)[O-])ccc2N1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PNMT P11086 5/20 0.42
ADRA2A P08913 3/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41
AR P10275 1/20 0.41
SIRT2 Q8IXJ6 1/20 0.40
ALDH1A1 P00352 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
SLC6A4 P31645 1/20 0.39
DRD3 P35462 1/20 0.39
OPRK1 P41145 1/20 0.39
HTR2B P41595 1/20 0.39
GRIN2B Q13224 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2776785 0.91 PNMT (0.43) PNMTADRA2AADRA2BADRA2CAR
SCHEMBL2778779 0.84 PNMT (0.46) PNMTADRA2AADRA2BADRA2CAR
SCHEMBL7456470 0.83 PNMT (0.56) PNMTADRA2AADRA2BADRA2CAR
SCHEMBL6195263 0.82 SIRT2 (0.45) PNMTADRA2AADRA2BADRA2CSIRT2
SCHEMBL2776959 0.81 ALDH1A1 (0.42) SIRT2ALDH1A1SMN1; SMN2GRIN2B
SCHEMBL6197463 0.81 PNMT (0.54) PNMTADRA2AADRA2BADRA2CSIRT2
SCHEMBL2775909 0.79 PNMT (0.33) PNMTADRA2AADRA2BADRA2CALDH1A1
SCHEMBL2776745 0.77 ALDH1A1 (0.41) PNMTSIRT2ALDH1A1SMN1; SMN2GRIN2B
SCHEMBL2857664 0.76 ALDH1A1 (0.52) PNMTADRA2AADRA2BADRA2CSIRT2
Bicarbonate SCHEMBL8143271 0.74 MAPK1 (0.40) PNMTADRA2AADRA2BADRA2CALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2139886-A1 QUINOLONE AND TETRAHYDROQUINOLINE AND RELATED COMPOUNDS HAVING NOS INHIBITORY ACTIVITY Neuraxon Inc. (CA) 2010-01-06 EP disclosed
WO-2008116308-A1 QUINOLONE AND TETRAHYDROQUINOLINE AND RELATED COMPOUNDS HAVING NOS INHIBITORY ACTIVITY NEURAXON, INC. (CA) 2008-10-02 WO disclosed