SCHEMBL27768216

SCHEMBL27768216

Cn1ncc(C(=O)O)c1Nc1ccccc1[N+](=O)[O-]

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 4/20 0.52
AKR1C2 P52895 4/20 0.52
KDM4E B2RXH2 2/20 0.52
ASPH Q12797 1/20 0.52
KDM8 Q8N371 1/20 0.52
MEN1 O00255 6/20 0.48
KMT2A Q03164 6/20 0.48
GAA P10253 3/20 0.48
MAPK1 P28482 3/20 0.48
TDP1 Q9NUW8 3/20 0.48
ALDH1A1 P00352 2/20 0.48
CASP7 P55210 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
POLB P06746 1/20 0.47
MAPT P10636 4/20 0.47
RAB9A P51151 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
AKR1B1 P15121 2/20 0.46
AKR1C4 P17516 2/20 0.46
AKR1C1 Q04828 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27789807 0.84 KCNMA1 (0.47) AKR1C3AKR1C2MEN1KMT2AGAA
SCHEMBL1496043 0.84 ALDH1A1 (0.48) MEN1KMT2AGAAMAPK1TDP1
SCHEMBL30933991 0.84 ALDH1A1 (0.48) MEN1KMT2AGAAMAPK1TDP1
SCHEMBL1495983 0.83 L3MBTL1 (0.50) AKR1C3AKR1C2MEN1KMT2AALDH1A1
SCHEMBL27789698 0.82 MEN1 (0.41) AKR1C3AKR1C2MEN1KMT2AGAA
SCHEMBL27540751 0.81 KDM4E (0.48) AKR1C3AKR1C2KDM4EASPHKDM8
SCHEMBL29989671 0.80 MAPK1 (0.47) KDM4EASPHKDM8MEN1KMT2A
SCHEMBL21378896 0.80 MAPK1 (0.47) KDM4EASPHKDM8MEN1KMT2A
SCHEMBL1495855 0.79 CDC25B (0.46) KDM4EMEN1KMT2AGAAMAPK1
SCHEMBL5554094 0.79 CDC25B (0.45) MEN1KMT2AGAAMAPK1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102617580-B Vasopressin v1a antagonists VANTIA LTD 2015-03-04 CN disclosed
CN-102617580-A Vasopressin V1a Antagonists FERRING BV 2012-08-01 CN disclosed
CN-101563347-A Vasopressin V1a antagonists VANTIA LTD (GB) 2009-10-21 CN disclosed