SCHEMBL3418996

SCHEMBL3418996

NNC(=O)c1nc(-c2cccnc2)no1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.57
KDM4E B2RXH2 2/20 0.56
CHRNB2 P17787 1/20 0.55
CHRNA5 P30532 1/20 0.55
CHRNA4 P43681 1/20 0.55
GSK3B P49841 10/20 0.54
MAPT P10636 3/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
HDAC1 Q13547 1/20 0.51
HDAC2 Q92769 1/20 0.51
HDAC8 Q9BY41 1/20 0.51
CA9 Q16790 1/20 0.50
PPARA Q07869 1/20 0.50
NPC1 O15118 1/20 0.50
ALDH1A1 P00352 1/20 0.50
TP53 P04637 1/20 0.50
HPGD P15428 1/20 0.50
RAB9A P51151 1/20 0.50
HSD17B10 Q99714 1/20 0.50
PIM1 P11309 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1432036 0.86 MKNK1 (0.57) KDM4ECHRNB2CHRNA5CHRNA4GSK3B
SCHEMBL2563085 0.84 GAA (0.68) GAAKDM4EMAPTNPC1ALDH1A1
SCHEMBL27768478 0.84 CHRNB2 (0.63) KDM4ECHRNB2CHRNA5CHRNA4MAPT
SCHEMBL1815822 0.82 CHRNB2 (0.61) KDM4ECHRNB2CHRNA5CHRNA4MAPT
SCHEMBL3419014 0.77 NPC1 (0.52) KDM4ECHRNB2CHRNA5CHRNA4MAPT
SCHEMBL7659667 0.77 HTT (0.60) KDM4ECHRNB2CHRNA5CHRNA4MAPT
SCHEMBL15639585 0.76 FAAH (0.56) GAAKDM4EMAPTSMN1; SMN2NPC1
SCHEMBL9233042 0.76 CHRNB2 (0.69) KDM4ECHRNB2CHRNA5CHRNA4MAPT
SCHEMBL14634348 0.75 GAA (0.68) GAAKDM4EMAPTSMN1; SMN2HDAC1
SCHEMBL22761300 0.75 CHRNB2 (0.63) KDM4ECHRNB2CHRNA5CHRNA4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593447-B1 3-PYRIDYL-HETEROARYLCARBOXAMIDE COMPOUNDS AS PESTICIDES BAYER IP GMBH (DE) 2016-08-17 EP disclosed
US-9233951-B2 Heterocyclic compounds as pesticides BAYER INTELLECTUAL PROPERTY GMBH (DE) 2016-01-12 US disclosed
US-9233951-B2 Heterocyclic compounds as pesticides BAYER INTELLECTUAL PROPERTY GMBH (DE) 2016-01-12 US disclosed
US-20120094837-A1 Novel Heterocyclic Compounds as Pesticides BAYER CROP SCIENCE AG (DE) 2012-04-19 US disclosed
US-20120094837-A1 Novel Heterocyclic Compounds as Pesticides BAYER CROP SCIENCE AG (DE) 2012-04-19 US disclosed
WO-2012007500-A2 NEW HETEROCYCLIC COMPOUNDS AS PESTICIDES BAYER CROPSCIENCE AG (DE) 2012-01-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120094837-A1 Novel Heterocyclic Compounds as Pesticides DDT, PTMS, ACHE GAA 2414/4885KDM4E 1038/4885CHRNB2 1540/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.