SCHEMBL27768691

SCHEMBL27768691

O=Cc1nc(-c2cccnc2)co1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.47
CYP2E1 P05181 2/20 0.47
CYP2C9 P11712 2/20 0.47
CYP2B6 P20813 2/20 0.47
CYP2C19 P33261 2/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2A6 P11509 5/20 0.45
ALDH1A1 P00352 3/20 0.45
CYP1A2 P05177 2/20 0.45
CYP19A1 P11511 4/20 0.45
AXL P30530 1/20 0.42
PBRM1 Q86U86 1/20 0.42
MKNK1 Q9BUB5 1/20 0.42
MKNK2 Q9HBH9 1/20 0.42
HSP90AA1 P07900 1/20 0.42
HSP90AB1 P08238 1/20 0.42
PTK2 Q05397 1/20 0.42
ERN1 O75460 1/20 0.42
METAP2 P50579 1/20 0.41
SIRT3 Q9NTG7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27768495 0.82 HSD11B1 (0.45) ALDH1A1RAB9AMAPTHPGDSMN1; SMN2
SCHEMBL15062621 0.81 CES1 (0.38) CYP3A4CYP2C9CYP2C19CYP2D6CYP1A2
SCHEMBL9346559 0.76 CYP2A6 (0.54) CYP3A4CYP2E1CYP2C9CYP2B6CYP2C19
SCHEMBL13984428 0.76 HSP90AA1 (0.53) CYP3A4CYP2E1CYP2C9CYP2B6CYP2C19
SCHEMBL6194452 0.73 CYP3A4 (0.55) CYP3A4CYP2E1CYP2C9CYP2B6CYP2C19
SCHEMBL27768689 0.73 CYP2A6 (0.45) CYP3A4CYP2A6ALDH1A1CYP1A2CYP19A1
SCHEMBL6821852 0.72 HDAC1 (0.37) ALDH1A1METAP2NPC1RAB9AKDM4E
SCHEMBL24623245 0.72 ADRB2 (0.50) CYP3A4CYP2E1CYP2C9CYP2B6CYP2C19
SCHEMBL4376192 0.72 RAB9A (0.65) ALDH1A1NPC1RAB9AKDM4ETP53
SCHEMBL28756282 0.72 MKNK1 (0.50) CYP3A4CYP2A6ALDH1A1CYP1A2CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102850324-A Indole compounds MICROBIA INC 2013-01-02 CN disclosed
CN-101563337-A Indole compounds MICROBIA INC (US) 2009-10-21 CN disclosed