SCHEMBL27768689

SCHEMBL27768689

O=C(c1nc(-c2cccnc2)co1)c1nc(-c2cccnc2)co1

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 4/20 0.45
CYP3A4 P08684 2/20 0.45
ALDH1A1 P00352 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP19A1 P11511 3/20 0.45
CES1 P23141 1/20 0.44
MKNK1 Q9BUB5 3/20 0.44
MKNK2 Q9HBH9 3/20 0.44
DAGLA Q9Y4D2 1/20 0.43
AXL P30530 1/20 0.42
PBRM1 Q86U86 1/20 0.42
HSP90AA1 P07900 1/20 0.42
HSP90AB1 P08238 1/20 0.42
PTK2 Q05397 1/20 0.42
IKBKB O14920 1/20 0.42
KMO O15229 2/20 0.42
METAP2 P50579 1/20 0.41
SIRT3 Q9NTG7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28756282 0.89 MKNK1 (0.50) CYP2A6CYP3A4ALDH1A1CYP1A2CYP19A1
SCHEMBL27768494 0.82 DAGLA (0.57) ALDH1A1CES1DAGLA
SCHEMBL27768589 0.81 CES1 (0.53) ALDH1A1CES1DAGLA
SCHEMBL13984428 0.76 HSP90AA1 (0.53) CYP2A6CYP3A4ALDH1A1CYP1A2CYP19A1
SCHEMBL9346559 0.76 CYP2A6 (0.54) CYP2A6CYP3A4ALDH1A1CYP1A2CYP19A1
SCHEMBL27605054 0.73 KMO (0.49) CYP2A6CYP3A4ALDH1A1CYP1A2CYP19A1
SCHEMBL27768691 0.73 CYP3A4 (0.47) CYP2A6CYP3A4ALDH1A1CYP1A2CYP19A1
SCHEMBL3199709 0.73 FAAH (0.70) CES1DAGLA
SCHEMBL24623245 0.72 ADRB2 (0.50) CYP2A6CYP3A4ALDH1A1CYP1A2CYP19A1
SCHEMBL27768478 0.72 CHRNB2 (0.63) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102850324-A Indole compounds MICROBIA INC 2013-01-02 CN disclosed
CN-101563337-A Indole compounds MICROBIA INC (US) 2009-10-21 CN disclosed