SCHEMBL28756282

SCHEMBL28756282

O=C(O)c1nc(-c2cccnc2)co1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 2/20 0.50
MKNK2 Q9HBH9 2/20 0.50
KMO O15229 2/20 0.48
CYP19A1 P11511 2/20 0.47
CES1 P23141 1/20 0.46
PIM1 P11309 1/20 0.46
PIM2 Q9P1W9 1/20 0.46
DAGLA Q9Y4D2 1/20 0.45
ALDH1A1 P00352 3/20 0.44
APP P05067 1/20 0.44
GAA P10253 1/20 0.44
HCAR3 P49019 1/20 0.44
HCAR2 Q8TDS4 1/20 0.44
CYP2A6 P11509 3/20 0.44
KDM4E B2RXH2 2/20 0.44
LMNA P02545 2/20 0.44
HTT P42858 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
DHODH Q02127 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27768689 0.89 CYP2A6 (0.45) MKNK1MKNK2KMOCYP19A1CES1
SCHEMBL5296166 0.84 DAGLA (0.57) CES1DAGLAALDH1A1KDM4ELMNA
SCHEMBL30528382 0.75 HCAR2 (0.43) CES1PIM1PIM2DAGLAALDH1A1
SCHEMBL3718120 0.75 ENPP3 (0.54) KMODAGLAALDH1A1KDM4EDHODH
SCHEMBL9346559 0.75 CYP2A6 (0.54) MKNK1MKNK2CYP19A1ALDH1A1CYP2A6
SCHEMBL13984428 0.75 HSP90AA1 (0.53) MKNK1MKNK2CYP19A1ALDH1A1GAA
SCHEMBL363026 0.74 KMO (0.59) MKNK1MKNK2KMOCYP19A1PIM1
SCHEMBL27768494 0.74 DAGLA (0.57) CES1DAGLAALDH1A1RAB9A
SCHEMBL1815822 0.73 CHRNB2 (0.61) MKNK1MKNK2ALDH1A1KDM4ELMNA
SCHEMBL12571348 0.73 ALDH1A1 (0.54) MKNK1MKNK2KMOPIM1PIM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1774435-A 5-membered heterocyclic derivative DAIICHI SEIYAKU CO (JP) 2006-05-17 CN disclosed