SCHEMBL27787296

SCHEMBL27787296

CN1c2ccccc2C(C=O)CS1(=O)=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 2/20 0.32
HTR6 P50406 2/20 0.32
POLB P06746 1/20 0.32
NOTUM Q6P988 1/20 0.31
HDAC4 P56524 1/20 0.31
HDAC7 Q8WUI4 1/20 0.31
HDAC5 Q9UQL6 1/20 0.31
GPR3 P46089 1/20 0.31
HTR2A P28223 2/20 0.31
LMNA P02545 2/20 0.31
MEN1 O00255 2/20 0.31
TP53 P04637 2/20 0.31
CYP1A2 P05177 2/20 0.31
CYP3A4 P08684 2/20 0.31
CYP2C9 P11712 2/20 0.31
CYP2C19 P33261 2/20 0.31
KMT2A Q03164 2/20 0.31
SLC6A2 P23975 2/20 0.31
SLC6A4 P31645 2/20 0.31
HTT P42858 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29243638 0.77 AADAT (0.38) HRH1POLBNOTUMHDAC4HDAC7
SCHEMBL14051069 0.73 MTNR1A (0.38) HRH1HTR6NOTUMHDAC4HDAC7
SCHEMBL27500006 0.70 KDM4C (0.38) HRH1HTR6NOTUMHDAC4HDAC7
SCHEMBL27716440 0.65 MAPT (0.39)
SCHEMBL14543698 0.65 NOTUM (0.64) NOTUMHTR2AHTTHTR1ADRD2
SCHEMBL28780260 0.64 OPRM1 (0.37) HTR6DRD2OPRM1DRD3OPRK1
SCHEMBL8264301 0.64 CACNA1G (0.33) NOTUMLMNAKDM4EOPRM1
SCHEMBL19194596 0.63 CA2 (0.43) NOTUMCYP1A2CYP2C9CYP2C19HTT
SCHEMBL28119505 0.63 SLC6A2 (0.54) SLC6A2SLC6A4SLC6A3
SCHEMBL8261724 0.63 CYP2C9 (0.40) POLBLMNAMEN1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101605776-A 4-imidazolyl-1, 2,3, 4-tetrahydroquinoline derivatives and their use as aldosterone/11-beta-hydroxylase inhibitors NOVARTIS AG (CH) 2009-12-16 CN disclosed