SCHEMBL27797604

SCHEMBL27797604

Oc1cccc(C2C3CC4CC(C3)CC2C4)c1F

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.34
CHRNA4 P43681 2/20 0.34
SCN9A Q15858 2/20 0.33
KDM1A O60341 1/20 0.33
EPHX2 P34913 5/20 0.32
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
HTR2B P41595 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL345589 0.81 HTR2A (0.42) CHRNB2CHRNA4SCN9AEPHX2HTR2A
SCHEMBL7745693 0.80 CHRNB2 (0.42) CHRNB2CHRNA4SCN9AHTR2AHTR2C
SCHEMBL2710155 0.80 G6PD (0.36) CHRNB2CHRNA4SCN9AHTR2AHTR2C
SCHEMBL15531515 0.79 TRPA1 (0.41) CHRNB2CHRNA4SCN9AEPHX2HTR2A
SCHEMBL5365399 0.75 SMN1; SMN2 (0.38) KDM1AEPHX2HTR2AHTR2CHTR2B
SCHEMBL27520667 0.75 CHRNB2 (0.39) CHRNB2CHRNA4SCN9AEPHX2
SCHEMBL15531513 0.71 ALDH1A1 (0.45) SCN9AHTR2AHTR2CHTR2B
SCHEMBL25981340 0.71 NOTUM (0.40) CHRNB2CHRNA4
SCHEMBL19249590 0.69 SCN9A (0.40) SCN9AEPHX2
SCHEMBL4614491 0.69 SCN9A (0.34) CHRNB2CHRNA4SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107501099-A The adjusting control agent of ATP combination cassette transporters 沃泰克斯药物股份有限公司 2017-12-22 CN disclosed
CN-104788328-B The adjusting control agent of ATP combination cassette transporters 沃泰克斯药物股份有限公司 2017-09-12 CN disclosed
CN-101935301-A Modulators of ATP-binding cassette transporters VERTEX PHARMA 2011-01-05 CN disclosed
CN-101891680-A The adjusting control agent of ATP- combination cassette transporters VERTEX PHARMA 2010-11-24 CN disclosed