SCHEMBL2789762

SCHEMBL2789762

CC(=O)NCCn1c(C2CCCN(C(=O)C[C@@H](Cc3ccc(B4OC(C)(C)C(C)(C)O4)cc3)NC(=O)O)C2)cc2c(Cl)cccc21

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 2/20 0.31
ITGA4 P13612 2/20 0.31
ITGB3 P05106 1/20 0.31
ITGA2B P08514 1/20 0.31
TACR2 P21452 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2790508 0.88 FPR2 (0.34) ITGB1ITGA4ITGB3ITGA2BKDM4E
SCHEMBL2791052 0.88 PROKR1 (0.34)
SCHEMBL2814040 0.82 CNR2 (0.34) ALDH1A1
SCHEMBL2814043 0.82 CNR2 (0.34) ALDH1A1
SCHEMBL2790813 0.79 PROKR1 (0.36) ITGB3ITGA2BTACR2ALDH1A1
SCHEMBL2791994 0.78 DPP4 (0.38) KDM4EALDH1A1GAA
SCHEMBL2790320 0.77 KDM4E (0.42) ITGB3ITGA2BKDM4EALDH1A1
SCHEMBL2790479 0.76 ALDH1A1 (0.31) ALDH1A1
SCHEMBL2790483 0.76 ALDH1A1 (0.31) ALDH1A1
SCHEMBL7898296 0.75 CNR2 (0.33) ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111634-A2 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-30 WO disclosed