SCHEMBL23112352

SCHEMBL23112352

COc1ccc(C2(O)CN(C(=O)O)C2)cn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NNMT P40261 1/20 0.42
GRIN2B Q13224 1/20 0.39
SCN9A Q15858 1/20 0.39
MKNK1 Q9BUB5 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38
ALDH1A1 P00352 3/20 0.38
GPR183 P32249 2/20 0.38
KMT2A Q03164 4/20 0.37
MEN1 O00255 3/20 0.37
KDM4E B2RXH2 2/20 0.37
MAPT P10636 1/20 0.37
POLB P06746 1/20 0.36
CCR2 P41597 2/20 0.36
BACE1 P56817 1/20 0.36
OPRM1 P35372 1/20 0.36
OPRL1 P41146 1/20 0.36
NPC1 O15118 1/20 0.36
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2790975 0.89 ALDH1A1 (0.40) NNMTGRIN2BSCN9AALDH1A1GPR183
SCHEMBL3662100 0.86 LMNA (0.43) NNMTGRIN2BALDH1A1KMT2AMEN1
SCHEMBL28548511 0.83 GPR119 (0.49) NNMTALDH1A1POLBBACE1HTT
SCHEMBL29977161 0.83 GPR119 (0.49) NNMTALDH1A1POLBBACE1HTT
SCHEMBL23112901 0.79 NNMT (0.37) NNMTSCN9AMKNK1MKNK2ALDH1A1
SCHEMBL23112557 0.79 OPRD1 (0.39) NNMTGRIN2BSCN9AGPR183KMT2A
SCHEMBL16874757 0.77 OPRM1 (0.48) GRIN2BALDH1A1KMT2AMEN1MAPT
SCHEMBL3469434 0.76 GPR119 (0.48) BACE1
SCHEMBL23231746 0.75 NNMT (0.41) NNMTSCN9AMKNK1MKNK2ALDH1A1
SCHEMBL23647652 0.75 NNMT (0.43) NNMTMKNK1MKNK2ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3793559-A1 SUBSTITUTED DIHYDROPYRAZOLO PYRAZINE CARBOXAMIDE DERIVATIVES Bayer Aktiengesellschaft (DE) 2021-03-24 EP disclosed