SCHEMBL27927691

SCHEMBL27927691

O=C1Nc2cc(Cl)cc(Cl)c2C1(O)C(F)(F)F

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
TP53 P04637 2/20 0.45
MAPT P10636 2/20 0.45
ALOX12 P18054 1/20 0.42
CES1 P23141 1/20 0.40
PDK2 Q15119 2/20 0.39
HTR6 P50406 7/20 0.38
DRD1 P21728 1/20 0.38
AR P10275 5/20 0.37
PKM P14618 1/20 0.36
GHSR Q92847 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27945952 0.79 ALDH1A1 (0.39) ALDH1A1TP53MAPTALOX12CES1
SCHEMBL5981551 0.67 ALDH1A1 (0.47) ALDH1A1TP53MAPTALOX12HTR6
SCHEMBL6180564 0.65 ALDH1A1 (0.46) ALDH1A1TP53MAPTALOX12HTR6
SCHEMBL733450 0.65 ALDH1A1 (0.58) ALDH1A1TP53MAPTALOX12HTR6
SCHEMBL3459900 0.65 HTR6 (0.55) ALDH1A1TP53MAPTHTR6DRD1
SCHEMBL128252 0.65 HTR6 (0.51) ALDH1A1TP53MAPTHTR6DRD1
SCHEMBL1770690 0.64 LCAT (0.36) AR
SCHEMBL5982243 0.64 KCNQ3 (0.46) ALDH1A1TP53MAPTALOX12HTR6
SCHEMBL24898308 0.63 POLB (0.34) PDK2PKM
SCHEMBL30211424 0.63 POLB (0.34) PDK2PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103443076-B Indol-2-one derivatives disubstituted in position 3, their preparation and their therapeutic application 赛诺菲-安万特 2016-06-22 CN disclosed
CN-103443076-A Indol-2-one derivatives disubstituted in position 3, their preparation and their therapeutic application SANOFI AVENTIS 2013-12-11 CN disclosed