SCHEMBL28004642

SCHEMBL28004642

c1ccc(CC2=NCCS2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.43
LMNA P02545 2/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2D6 P10635 2/20 0.43
POLB P06746 1/20 0.43
ADRA2A P08913 1/20 0.43
TSHR P16473 1/20 0.43
ADRA2B P18089 1/20 0.43
ADRA2C P18825 1/20 0.43
ADRA1D P25100 1/20 0.43
ADRA1A P35348 1/20 0.43
ADRA1B P35368 1/20 0.43
CALM1 P0DP23 1/20 0.42
SORT1 Q99523 1/20 0.41
TP53 P04637 2/20 0.40
ALDH1A1 P00352 5/20 0.39
NPSR1 Q6W5P4 1/20 0.39
RAB9A P51151 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
TDP1 Q9NUW8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20746327 0.80 CHRNB2 (0.43) LMNACYP1A2CYP2D6TP53ALDH1A1
SCHEMBL3290862 0.69 GFER (0.60) LMNACYP2D6ALDH1A1RAB9ASMN1; SMN2
Bromide SCHEMBL6206034 0.68 TP53 (0.53) CYP1A2CYP2D6TP53ALDH1A1RAB9A
SCHEMBL1147751 0.68 LMNA (0.53) TAAR1LMNAPOLBTP53ALDH1A1
Hydrochloric Acid SCHEMBL4211382 0.67 ALDH1A1 (0.56) TAAR1LMNAPOLBTSHRTP53
SCHEMBL17831415 0.66 EPHX1 (0.42) TAAR1LMNACYP1A2CYP2D6POLB
SCHEMBL2017733 0.66 ALDH1A1 (0.82) TAAR1LMNAPOLBTSHRTP53
SCHEMBL8726368 0.65 CALM1 (0.39) TAAR1LMNACYP1A2CYP2D6POLB
SCHEMBL697719 0.65 TAAR1 (0.44) TAAR1LMNACYP1A2CYP2D6POLB
SCHEMBL2665231 0.64 CALM1 (0.38) TAAR1LMNACYP1A2CYP2D6ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106032365-B Benzal thiazolinone of 2 (base of thiazole 2) imino group 5 and preparation method and application 湖南大学 2018-03-23 CN disclosed
CN-105985298-A 2-[5-(halogenothiazolyl-2-yl)imino]-5-benzalthiazolinone and its preparation method and use 湖南大学 2016-10-05 CN disclosed
CN-103304507-B Green method for preparing heterocyclic compounds from nitriles UNIV WENZHOU 2015-02-25 CN disclosed