SCHEMBL1147751

SCHEMBL1147751

c1ccc(C2=NCCS2)cc1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
POLB P06746 1/20 0.47
ALDH1A1 P00352 2/20 0.45
MAPT P10636 1/20 0.45
ATM Q13315 1/20 0.45
TAAR1 Q96RJ0 1/20 0.41
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
CASP3 P42574 1/20 0.40
SENP8 Q96LD8 1/20 0.40
SENP7 Q9BQF6 1/20 0.40
SENP6 Q9GZR1 1/20 0.40
TP53 P04637 1/20 0.40
MGLL Q99685 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27368504 0.86 LMNA (0.58) LMNASMN1; SMN2POLBALDH1A1MAPT
SCHEMBL21663870 0.80 MAPT (0.48) LMNASMN1; SMN2ALDH1A1MAPTATM
SCHEMBL20411019 0.78 ALDH1A1 (0.43) LMNASMN1; SMN2ALDH1A1MAPTATM
SCHEMBL8378973 0.78 MGLL (0.43) LMNASMN1; SMN2ALDH1A1MAPTATM
SCHEMBL21664123 0.78 ALDH1A1 (0.47) LMNASMN1; SMN2ALDH1A1MAPTATM
SCHEMBL5777989 0.78 ALDH1A1 (0.43) LMNASMN1; SMN2ALDH1A1MAPTATM
SCHEMBL6170485 0.78 CYP2A6 (0.50) LMNASMN1; SMN2ALDH1A1MAPTATM
SCHEMBL27886244 0.77 ALDH1A1 (0.60) LMNASMN1; SMN2ALDH1A1MAPTATM
SCHEMBL27605025 0.77 LMNA (0.56) LMNASMN1; SMN2ALDH1A1
SCHEMBL28434848 0.77 SMN1; SMN2 (0.49) LMNASMN1; SMN2ALDH1A1MAPTATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 62 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100404540-C Thiazolo-, oxazolo-and imidazoquinazoline compounds which inhibit protein kinases CYCLACEL LTD (GB) 2008-07-23 CN claimed
CN-1849325-A Thiazolo-, oxazalo and imidazolo-quinazoline compounds capable of inhibiting prot ein kinases CYCLACEL LTD (GB) 2006-10-18 CN claimed
US-6955921-B2 Trypsin substrate and diagnostic device, and method of using same BAYER CORPORATION (US) 2005-10-18 US claimed
EP-1529037-A2 SYNTHESIS OF 2-ALKYLCYSTEINES, 2-(HYDROXYLATED PHENYL)-4-ALKYLTHIAZOLINE-4-CARBOXYLIC ACIDS AND DERIVATIVES THEREOF Genzyme Corporation (US) 2005-05-11 EP claimed
US-6770764-B2 DIAGNOSIS OF BACTERIA INFECTIONS BAYER CORPORATION 2004-08-03 US claimed
US-20030236404-A1 Synthesis of 2-alkylcysteine via phase transfer catalysis GENZYME CORPORATION 2003-12-25 US claimed
WO-2003097622-A2 SYNTHESIS OF 2-ALKYLCYSTEINES, 2-(HYDROXYLATED PHENYL)-4-ALKYLTHIAZOLINE-4-CARBOXYLIC ACIDS AND DERIVATIVES THEREOF GENZYME CORPORATION (US) 2003-11-27 WO claimed
US-20030125577-A1 Trypsin substrate and diagnostic device, and method of using same SIEMENS HEALTHCARE DIAGNOSTICS INC. 2003-07-03 US claimed
US-20020004219-A1 Trypsin substrate and diganostic device, and method of using same SIEMENS HEALTHCARE DIAGNOSTICS INC. 2002-01-10 US claimed
EP-1157984-A2 Trypsin substrate and diagnostic device, and method of using same Bayer Corporation (US) 2001-11-28 EP claimed
EP-0432661-B1 2-Substituted phenyl-2-oxazoline or thiazoline derivatives, process for producing the same and insecticides and acaricides containing the same YASHIMA KAGAKU KOGYO KK (JP) 1996-03-06 EP claimed
EP-0432661-A2 2-Substituted phenyl-2-oxazoline or thiazoline derivatives, process for producing the same and insecticides and acaricides containing the same YASHIMA CHEMICAL INDUSTRIAL CO., LTD. (JP) 1991-06-19 EP claimed
CN-119776090-A Soft endoscope strong-effect multienzyme cleaning agent and preparation process thereof 杭州西子卫生消毒药械有限公司 2025-04-08 CN disclosed
CN-114805348-A Triazolopyridine amide compound and preparation method and application thereof 贵州大学 2022-07-29 CN disclosed
US-11342511-B2 Azoline ring-containing compound, electron transport/injection layer material containing the same, and organic electroluminescent element using the same SK MATERIALS JNC CO., LTD. (KR) 2022-05-24 US disclosed
US-11319347-B2 Peptide compound and method for producing same, composition for screening use, and method for selecting peptide compound FUJIFILM CORPORATION (JP) 2022-05-03 US disclosed
EP-0203359-A2 Novel peptide having dentinal fluid transport stimulating activity TEIKOKU HORMONE MFG. CO., LTD. (JP) 1986-12-03 EP disclosed
EP-0132165-A1 Adsorbable alkynyl substituted heterocyclic quaternary ammonium salts and applications thereof to silver halide photography EASTMAN KODAK COMPANY (a New Jersey corporation) (US) 1985-01-23 EP disclosed
US-4471044-A Silver halide emulsions and photographic elements containing adsorbable alkynyl substituted heterocyclic quaternary ammonium salts EASTMAN KODAK COMPANY (US) 1984-09-11 US disclosed
US-4115122-A Internal latent image silver halide emulsion containing a heterocyclic quaternary salt having a propargyl or a butyryl containing substituent FUJI PHOTO FILM CO., LTD. (JP) 1978-09-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020004219-A1 Trypsin substrate and diganostic device, and method of using same PRSS3, CTRL, PRSS2 LMNA 1790/4885SMN1; SMN2 4365/4885POLB 2537/4885
US-20030236404-A1 Synthesis of 2-alkylcysteine via phase transfer catalysis DIMT1, ICMT, CNDP2 LMNA 4323/4885SMN1; SMN2 2739/4885POLB 4039/4885
US-11342511-B2 Azoline ring-containing compound, electron transport/injection layer material containing the same, and organic electroluminescent element using the same SLC7A5, EML4, ARNT LMNA 1407/4885SMN1; SMN2 3753/4885POLB 3289/4885
US-11319347-B2 Peptide compound and method for producing same, composition for screening use, and method for selecting peptide compound VIP, NPPA, NGLY1 LMNA 3026/4885SMN1; SMN2 3728/4885POLB 4749/4885
US-20030125577-A1 Trypsin substrate and diagnostic device, and method of using same CTRL, PRSS3, SPINT2 LMNA 1936/4885SMN1; SMN2 3309/4885POLB 2333/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.