SCHEMBL28007656

SCHEMBL28007656

COCCCc1c[nH]c2cc(C(=O)O)ncc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.40
MTNR1A P48039 8/20 0.40
MTNR1B P49286 8/20 0.40
NPC1 O15118 1/20 0.38
PRKAB2 O43741 1/20 0.37
PRKAG1 P54619 1/20 0.37
PRKAA2 P54646 1/20 0.37
PRKAA1 Q13131 1/20 0.37
PRKAG3 Q9UGI9 1/20 0.37
PRKAG2 Q9UGJ0 1/20 0.37
PRKAB1 Q9Y478 1/20 0.37
TRPV1 Q8NER1 1/20 0.36
CYP1A2 P05177 3/20 0.36
CYP3A4 P08684 3/20 0.36
CYP2D6 P10635 3/20 0.36
KMT2A Q03164 2/20 0.36
KDM4E B2RXH2 1/20 0.36
HPGD P15428 1/20 0.36
APEX1 P27695 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL28007658 0.99 HCAR2 (0.39) HCAR2MTNR1AMTNR1BNPC1PRKAB2
SCHEMBL28007337 0.85 GABRG2 (0.43) MTNR1AMTNR1BNPC1
SCHEMBL16610221 0.79 MTNR1B (0.38) MTNR1AMTNR1BKMT2AMEN1SLC6A4
SCHEMBL4915074 0.73 GABRA1 (0.46) NPC1CYP1A2CYP3A4CYP2D6KDM4E
SCHEMBL28819880 0.72 GABRA1 (0.46) MTNR1AMTNR1BNPC1CYP1A2CYP3A4
SCHEMBL1046830 0.71 MTNR1B (0.45) MTNR1AMTNR1BCYP1A2CYP3A4CYP2D6
SCHEMBL18080758 0.70 MTNR1B (0.39) MTNR1AMTNR1BNPC1CYP1A2CYP2D6
SCHEMBL1050599 0.69 MTNR1A (0.43) MTNR1AMTNR1BCYP3A4CYP2C9CYP2C19
SCHEMBL19555767 0.68 HCAR2 (0.42) HCAR2CYP1A2CYP3A4KMT2AKDM4E
SCHEMBL30112008 0.68 HCAR2 (0.42) HCAR2CYP1A2CYP3A4KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104640847-B Novel Renin Inhibitors 上海医药集团股份有限公司 2019-10-15 CN disclosed
CN-104640847-A Novel Renin Inhibitors SHANGHAI PHARMACEUTICALS HOLDING CO LTD 2015-05-20 CN disclosed