SCHEMBL28007337

SCHEMBL28007337

COCCCc1c[nH]c2cc(C(=O)OC(C)(C)C)ncc12

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 13/20 0.43
GABRB3 P28472 13/20 0.43
GABRA1 P14867 12/20 0.43
GABRA2 P47869 12/20 0.43
GABRA5 P31644 12/20 0.43
GABRA3 P34903 11/20 0.43
GABRA6 Q16445 10/20 0.43
GABRA4 P48169 5/20 0.43
GABRP O00591 1/20 0.43
GABRD O14764 1/20 0.43
GABRB1 P18505 1/20 0.43
GABRB2 P47870 1/20 0.43
GABRE P78334 1/20 0.43
GABRG1 Q8N1C3 1/20 0.43
GABRG3 Q99928 1/20 0.43
GABRQ Q9UN88 1/20 0.43
NPC1 O15118 1/20 0.37
MTNR1A P48039 2/20 0.36
MTNR1B P49286 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28007656 0.85 HCAR2 (0.40) NPC1MTNR1AMTNR1B
Hydrochloric Acid SCHEMBL28007658 0.84 HCAR2 (0.39) NPC1MTNR1AMTNR1B
SCHEMBL2806960 0.76 GABRG2 (0.50) GABRG2GABRB3GABRA1GABRA2GABRA5
SCHEMBL16610221 0.74 MTNR1B (0.38) MTNR1AMTNR1B
SCHEMBL4915074 0.74 GABRA1 (0.46) GABRG2GABRB3GABRA1GABRA2GABRA5
SCHEMBL28819880 0.73 GABRA1 (0.46) GABRG2GABRB3GABRA1GABRA2GABRA5
SCHEMBL18508705 0.69 GABRA1 (0.41) GABRG2GABRB3GABRA1GABRA2GABRA5
SCHEMBL2297259 0.68 GABRG2 (0.52) GABRG2GABRB3GABRA1GABRA2GABRA5
SCHEMBL12526818 0.67 REN (0.44) GABRG2GABRB3GABRA1GABRA2GABRA5
SCHEMBL1046830 0.67 MTNR1B (0.45) MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104640847-B Novel Renin Inhibitors 上海医药集团股份有限公司 2019-10-15 CN disclosed
CN-104640847-A Novel Renin Inhibitors SHANGHAI PHARMACEUTICALS HOLDING CO LTD 2015-05-20 CN disclosed