SCHEMBL28021141

SCHEMBL28021141

Clc1cnn(-c2cccnc2)c1-c1cccnc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.46
PTGS2 P35354 1/20 0.46
CYP2A6 P11509 7/20 0.44
ALDH1A1 P00352 4/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP11B2 P19099 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
CHRNB2 P17787 1/20 0.42
CHRNA5 P30532 1/20 0.42
CHRNA4 P43681 1/20 0.42
KEAP1 Q14145 1/20 0.41
NFE2L2 Q16236 1/20 0.41
MAPT P10636 4/20 0.39
KDM4E B2RXH2 2/20 0.39
HTT P42858 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
GRM1 Q13255 1/20 0.39
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14747796 0.78 PTGS2 (0.68) PTGS1PTGS2ALDH1A1CYP1A2CYP3A4
SCHEMBL9026151 0.70 GRM1 (0.46) CYP2A6ALDH1A1CYP1A2CYP3A4CYP11B2
Sulfamide SCHEMBL7137771 0.70 PTGS2 (0.79) PTGS1PTGS2ALDH1A1MAPTHTT
SCHEMBL6237143 0.70 CYP11B2 (0.48) CYP2A6ALDH1A1CYP1A2CYP3A4CYP11B2
SCHEMBL15839004 0.70 CYP11B2 (0.48) CYP2A6ALDH1A1CYP3A4CYP11B2L3MBTL1
SCHEMBL15839181 0.70 CYP11B2 (0.48) CYP2A6CYP1A2CYP3A4CYP11B2GRM1
SCHEMBL6845949 0.68 CYP11B2 (0.68) CYP2A6ALDH1A1CYP1A2CYP3A4CYP11B2
SCHEMBL5731172 0.68 ALDH1A1 (0.46) PTGS1PTGS2CYP2A6ALDH1A1CYP1A2
SCHEMBL6157378 0.68 PTGS2 (0.63) PTGS1PTGS2ALDH1A1MAPTKDM4E
SCHEMBL6086847 0.66 CYP11B2 (0.46) CYP2A6CYP3A4CYP11B2L3MBTL1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104860927-A 1H-3,5-bis(3-pyridinyl)-4-chloropyrazole compound, and preparation method and application thereof UNIV NINGBO 2015-08-26 CN claimed