SCHEMBL28025014

SCHEMBL28025014

COC(=O)c1c(C(F)(F)F)[nH]c2ccc(OC(F)(F)F)cc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.51
CRHBP P24387 1/20 0.51
CRHR2 Q13324 1/20 0.51
KMT2A Q03164 2/20 0.44
GAA P10253 1/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
TRPV1 Q8NER1 4/20 0.43
KIF11 P52732 1/20 0.43
MEN1 O00255 1/20 0.42
MET P08581 1/20 0.41
PTGS2 P35354 2/20 0.41
CYP2C9 P11712 1/20 0.41
PTGS1 P23219 1/20 0.41
NR4A2 P43354 2/20 0.40
MAPT P10636 1/20 0.39
CCNT1 O60563 1/20 0.39
CCNE1 P24864 1/20 0.39
CDK2 P24941 1/20 0.39
CDK9 P50750 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19322278 0.91 NR4A2 (0.50) KDM4EKMT2AGAANPC1RAB9A
SCHEMBL28024552 0.90 KIF11 (0.49) KDM4ECRHBPCRHR2KMT2AGAA
SCHEMBL28207430 0.86 KDM4E (0.53) KDM4ECRHBPCRHR2KMT2AGAA
SCHEMBL28024557 0.84 NR4A2 (0.49) KDM4EKMT2AGAANPC1RAB9A
SCHEMBL28025008 0.83 ALOX5 (0.56) KDM4EKMT2AGAANPC1RAB9A
SCHEMBL28025005 0.82 RAB9A (0.52) KDM4EKMT2ANPC1RAB9AKIF11
SCHEMBL28206980 0.82 RAB9A (0.52) KDM4EKMT2ANPC1RAB9AKIF11
SCHEMBL28024558 0.81 NR4A2 (0.48) KDM4EKMT2AGAANPC1RAB9A
SCHEMBL19322108 0.80 ALDH1A1 (0.49) KDM4EKMT2AGAANPC1RAB9A
SCHEMBL28024553 0.80 KDM4E (0.54) KDM4EKMT2AGAANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105646327-A 2-perfluoroalkyl indole derivative and synthesis method thereof 上海大学 2016-06-08 CN disclosed
CN-104892485-A 2-perfluoroalkyl indole derivative and synthesis method thereof UNIV SHANGHAI 2015-09-09 CN disclosed