SCHEMBL28028735

SCHEMBL28028735

CC(=O)Nc1ccc2[nH]c(C(=O)NN)cc2c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 2/20 0.66
KDM4E B2RXH2 4/20 0.57
GAA P10253 2/20 0.57
ALDH1A1 P00352 1/20 0.57
MAPK1 P28482 1/20 0.57
HDAC2 Q92769 1/20 0.56
KMT2A Q03164 3/20 0.53
NPC1 O15118 2/20 0.50
RXFP1 Q9HBX9 2/20 0.50
RAB9A P51151 1/20 0.50
ROCK2 O75116 1/20 0.50
ROCK1 Q13464 1/20 0.50
TP53 P04637 2/20 0.49
POLB P06746 1/20 0.49
PLD2 O14939 1/20 0.48
PLD1 Q13393 1/20 0.48
NHERF1 O14745 1/20 0.48
PYGL P06737 1/20 0.48
EGFR P00533 2/20 0.48
PIK3CA P42336 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3027767 0.84 MMP13 (0.67) MMP13KDM4EALDH1A1KMT2AROCK2
SCHEMBL28028254 0.82 MAOA (0.66) KDM4EGAAALDH1A1MAPK1HDAC2
SCHEMBL22718557 0.81 PLD2 (0.56) KDM4EGAAALDH1A1MAPK1HDAC2
SCHEMBL28229577 0.80 TP53 (0.56) MMP13KDM4EHDAC2KMT2ANPC1
SCHEMBL28028262 0.80 MMP13 (0.59) MMP13KDM4EGAAHDAC2KMT2A
SCHEMBL28028261 0.80 MMP13 (0.59) MMP13KDM4EGAAHDAC2KMT2A
SCHEMBL6514040 0.80 MMP13 (1.00) MMP13KDM4EGAAALDH1A1KMT2A
SCHEMBL15746114 0.79 PIN1 (0.66) KDM4EGAAALDH1A1MAPK1HDAC2
SCHEMBL27520204 0.78 NPC1 (0.53) MMP13ALDH1A1MAPK1HDAC2KMT2A
SCHEMBL6015700 0.77 MAOB (0.67) MMP13KDM4EALDH1A1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104860866-B 5- (substitution carbon acylamino) -1H- indoles -2- carbohydrazide derivatives and its preparation method and application 厦门大学 2018-07-17 CN disclosed
CN-104860866-A 5-(substituted carbonylamino)-1H-indole-2-carbohydrazide derivatives as well as preparation method and application thereof UNIV XIAMEN 2015-08-26 CN disclosed