SCHEMBL28028254

SCHEMBL28028254

NNC(=O)c1cc2cc(NC(=O)c3ccccc3)ccc2[nH]1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.66
MAOB P27338 1/20 0.66
KDM4E B2RXH2 1/20 0.61
ALDH1A1 P00352 1/20 0.61
GAA P10253 1/20 0.61
MAPK1 P28482 1/20 0.61
EGFR P00533 5/20 0.61
PIK3CA P42336 5/20 0.61
TP53 P04637 1/20 0.59
POLB P06746 1/20 0.59
NPC1 O15118 3/20 0.58
RAB9A P51151 3/20 0.58
LMNA P02545 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
NHERF1 O14745 2/20 0.58
MAPT P10636 1/20 0.58
JAK2 O60674 1/20 0.55
HDAC2 Q92769 1/20 0.53
PIN1 Q13526 1/20 0.53
PYGL P06737 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10466165 0.88 MAOA (0.71) MAOAMAOBKDM4EALDH1A1EGFR
SCHEMBL22718557 0.85 PLD2 (0.56) MAOAMAOBKDM4EALDH1A1GAA
SCHEMBL28028277 0.85 MAOA (0.63) MAOAMAOBEGFRPIK3CATP53
SCHEMBL27325791 0.83 MAOA (0.60) MAOAMAOBALDH1A1EGFRPIK3CA
SCHEMBL28028735 0.82 MMP13 (0.66) KDM4EALDH1A1GAAMAPK1EGFR
SCHEMBL24601450 0.82 MMP13 (0.72) MAOAMAOBKDM4EALDH1A1GAA
SCHEMBL8205048 0.81 NHERF1 (0.64) MAOAMAOBKDM4EALDH1A1EGFR
SCHEMBL7533561 0.81 NPC1 (0.74) MAOAMAOBKDM4EEGFRPIK3CA
SCHEMBL27690981 0.81 MAOA (0.72) MAOAMAOBALDH1A1EGFRPIK3CA
SCHEMBL28028263 0.81 MAOA (0.58) MAOAMAOBKDM4EEGFRPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104860866-A 5-(substituted carbonylamino)-1H-indole-2-carbohydrazide derivatives as well as preparation method and application thereof UNIV XIAMEN 2015-08-26 CN claimed
CN-104860866-B 5- (substitution carbon acylamino) -1H- indoles -2- carbohydrazide derivatives and its preparation method and application 厦门大学 2018-07-17 CN disclosed
CN-104860866-A 5-(substituted carbonylamino)-1H-indole-2-carbohydrazide derivatives as well as preparation method and application thereof UNIV XIAMEN 2015-08-26 CN disclosed