SCHEMBL28036149

SCHEMBL28036149

COc1cc(N2CCN(C(=O)O)C(C(C)(C)C)C2)ccc1Br

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 2/20 0.40
LMNA P02545 2/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NR1H2 P55055 5/20 0.39
CHRM4 P08173 3/20 0.38
NR1H3 Q13133 3/20 0.38
CTSB P07858 2/20 0.37
CTSS P25774 2/20 0.37
CTSK P43235 2/20 0.37
ALK Q9UM73 1/20 0.37
CCR1 P32246 3/20 0.37
TRPC6 Q9Y210 1/20 0.35
SUV39H2 Q9H5I1 1/20 0.35
POLB P06746 1/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16752913 0.86 SLC6A9 (0.40) SLC6A9NR1H2CHRM4NR1H3CTSB
SCHEMBL3503419 0.83 SIRT6 (0.57) LMNAHTTSMN1; SMN2
SCHEMBL28036150 0.81 HTR1A (0.48) LMNAHTTSMN1; SMN2POLBGAA
SCHEMBL2442056 0.79 SLC6A9 (0.36) SLC6A9NR1H2CHRM4NR1H3CTSB
SCHEMBL17310201 0.79 SMN1; SMN2 (0.51) LMNAHTTSMN1; SMN2ALKCCR1
SCHEMBL11963285 0.79 NR1H2 (0.44) SMN1; SMN2NR1H2NR1H3
SCHEMBL26096595 0.79 HTR1D (0.37) LMNAHTTSMN1; SMN2TRPC6POLB
SCHEMBL26094770 0.78 LMNA (0.34) LMNAHTTSMN1; SMN2CHRM4TRPC6
SCHEMBL29252729 0.77 AGTR2 (0.48) NR1H2CHRM4NR1H3CTSBCTSS
SCHEMBL2760636 0.77 DRD2 (0.51) LMNASMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104968654-A Substituted 2-aminopyridine protein kinase inhibitor CHIA TAI TIANQING PHARMACEUTICAL GROUP CO LTD 2015-10-07 CN disclosed