SCHEMBL28041408

SCHEMBL28041408

COCCCOc1cc(C(C)C2[CH]C2)ccc1OCc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
REN P00797 10/20 0.49
C5AR1 P21730 5/20 0.40
ADRA1D P25100 4/20 0.39
ADRA1A P35348 4/20 0.39
ADRA1B P35368 4/20 0.39
HTR1A P08908 3/20 0.39
HTR2A P28223 2/20 0.38
HTR2B P41595 2/20 0.38
KCNH2 Q12809 2/20 0.38
KDM4E B2RXH2 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
F2 P00734 1/20 0.38
F10 P00742 1/20 0.38
PRSS1 P07477 1/20 0.38
PRSS2 P07478 1/20 0.38
F7 P08709 1/20 0.38
F3 P13726 1/20 0.38
PRSS3 P35030 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12524630 0.80 REN (0.50) RENC5AR1ADRA1DADRA1AADRA1B
SCHEMBL6943581 0.76 REN (0.47) RENC5AR1ADRA1DADRA1AADRA1B
SCHEMBL19526619 0.76 REN (0.59) RENADRA1DADRA1AADRA1BHTR1A
SCHEMBL28785298 0.76 MTNR1A (0.44) RENC5AR1KDM4E
SCHEMBL682767 0.76 MAPT (0.49) C5AR1KDM4ETDP1F2F10
SCHEMBL27795807 0.75 HTR1A (0.61) ADRA1DADRA1AADRA1BHTR1AKDM4E
SCHEMBL18715976 0.75 L3MBTL1 (0.52) C5AR1ADRA1DADRA1AADRA1BHTR1A
SCHEMBL13433963 0.75 L3MBTL1 (0.52) C5AR1ADRA1DADRA1AADRA1BHTR1A
SCHEMBL20577097 0.74 SIGMAR1 (0.47) RENADRA1DADRA1AADRA1B
SCHEMBL21042791 0.74 SLC6A4 (0.53) ADRA1DADRA1AADRA1BHTR1AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103562191-B Nitrogen-containing saturated heterocyclic compound SHANGHAI PHARMACEUTICALS HOLDING CO.,LTD. (CN) 2016-03-30 CN disclosed