SCHEMBL28044658

SCHEMBL28044658

O=C(O)c1cnc(C(F)(F)F)nc1I

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ASPH Q12797 2/20 0.41
ALDH1A1 P00352 1/20 0.37
KMT2A Q03164 1/20 0.37
FOS P01100 3/20 0.36
JUN P05412 3/20 0.36
NFKB1 P19838 3/20 0.36
NFKB2 Q00653 3/20 0.36
RELA Q04206 3/20 0.36
HPGD P15428 2/20 0.34
POLB P06746 1/20 0.34
MAPT P10636 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
PDE4B Q07343 4/20 0.34
KDM4E B2RXH2 2/20 0.33
KDM8 Q8N371 1/20 0.33
XPO1 O14980 1/20 0.33
TAS2R14 Q9NYV8 1/20 0.33
GABRP O00591 1/20 0.33
GABRD O14764 1/20 0.33
GABRA1 P14867 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8544671 0.80 XPO1 (0.42) ASPHALDH1A1KMT2AFOSJUN
SCHEMBL3283505 0.80 ASPH (0.42) ASPHALDH1A1KMT2AFOSJUN
SCHEMBL4415725 0.79 KEAP1 (0.44) ASPHALDH1A1KMT2AFOSJUN
SCHEMBL2352570 0.79 HPGD (0.53) ASPHALDH1A1KMT2AFOSJUN
SCHEMBL17393706 0.77 JUN (0.58) ALDH1A1KMT2AFOSJUNNFKB1
SCHEMBL18660845 0.75 HPGD (0.39) ASPHALDH1A1KMT2AHPGDPOLB
SCHEMBL22868013 0.75 POLB (0.46) ASPHALDH1A1KMT2AFOSJUN
SCHEMBL14809757 0.75 GABRP (0.45) ASPHALDH1A1KMT2AFOSJUN
SCHEMBL1759984 0.73 PDE4B (0.40) ASPHALDH1A1KMT2AFOSJUN
SCHEMBL15639612 0.72 CDK2 (0.46) FOSJUNNFKB1NFKB2RELA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105073715-B The derovatives of dihydrogen dazin 3,5 中外制药株式会社 2017-12-01 CN disclosed
CN-105073715-A Dihydropyridazine-3,5-dione derivative CHUGAI PHARMACEUTICAL CO LTD 2015-11-18 CN disclosed