SCHEMBL28044959

SCHEMBL28044959

O=C(Cc1cccc(O)c1)NCc1ccc(Br)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.70
MEN1 O00255 2/20 0.60
KMT2A Q03164 2/20 0.60
NLRP3 Q96P20 2/20 0.60
CA1 P00915 1/20 0.55
CA2 P00918 1/20 0.55
HSD17B2 P37059 1/20 0.55
ALDH1A1 P00352 4/20 0.51
ERCC1 P07992 2/20 0.51
ERCC4 Q92889 2/20 0.51
LMNA P02545 1/20 0.51
ROS1 P08922 1/20 0.50
RPS6KB1 P23443 1/20 0.50
RAB9A P51151 1/20 0.50
HDAC3 O15379 1/20 0.50
HDAC4 P56524 1/20 0.50
HDAC1 Q13547 1/20 0.50
HDAC7 Q8WUI4 1/20 0.50
HDAC2 Q92769 1/20 0.50
HDAC10 Q969S8 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16747758 0.88 CA1 (0.64) L3MBTL1MEN1KMT2ANLRP3CA1
SCHEMBL1656898 0.83 L3MBTL1 (1.00) L3MBTL1MEN1KMT2ACA1CA2
SCHEMBL5177163 0.82 NLRP3 (0.62) NLRP3CA1CA2HSD17B2LMNA
SCHEMBL26625402 0.82 NLRP3 (0.62) NLRP3CA1CA2HSD17B2ALDH1A1
SCHEMBL1748615 0.78 ALDH1A1 (0.75) L3MBTL1MEN1KMT2ANLRP3CA1
SCHEMBL13199178 0.78 NPC1 (0.55) L3MBTL1MEN1KMT2ANLRP3ALDH1A1
SCHEMBL2810721 0.78 SRC (0.73) L3MBTL1MEN1KMT2AALDH1A1ERCC1
SCHEMBL24439952 0.78 NLRP3 (0.64) L3MBTL1MEN1KMT2ANLRP3CA1
SCHEMBL29605976 0.78 NLRP3 (0.64) L3MBTL1MEN1KMT2ANLRP3CA1
SCHEMBL8480688 0.76 PKM (0.53) KMT2ANLRP3ERCC1ERCC4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105294458-A Antineoplastic small molecular compound and preparation method and application thereof FOURTH MILITARY MEDICAL UNIV 2016-02-03 CN claimed
CN-105294458-B A kind of anti-tumor small molecular compound and its preparation method and application 中国人民解放军第四军医大学 2017-07-11 CN disclosed
CN-105294458-A Antineoplastic small molecular compound and preparation method and application thereof FOURTH MILITARY MEDICAL UNIV 2016-02-03 CN disclosed
CN-105294458-A Antineoplastic small molecular compound and preparation method and application thereof FOURTH MILITARY MEDICAL UNIV 2016-02-03 CN disclosed