SCHEMBL28045207

SCHEMBL28045207

CC(=O)OC(C)Oc1ccc(N)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.42
PARP10 Q53GL7 2/20 0.42
POLB P06746 1/20 0.40
TDP1 Q9NUW8 5/20 0.39
TSHR P16473 3/20 0.39
KMT2A Q03164 1/20 0.39
MAPK1 P28482 1/20 0.39
GLA P06280 1/20 0.39
ALDH1A1 P00352 3/20 0.38
CYP3A4 P08684 2/20 0.38
NPC1 O15118 1/20 0.36
TP53 P04637 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CYP1A2 P05177 1/20 0.36
GAA P10253 1/20 0.36
CYP2C9 P11712 1/20 0.36
PKM P14618 1/20 0.36
CYP2C19 P33261 1/20 0.36
TAS1R3 Q7RTX0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10063720 0.90 POLB (0.46) PARP10POLBTDP1TSHRKMT2A
SCHEMBL13763456 0.83 LMNA (0.53) PARP10POLBTDP1TSHRKMT2A
SCHEMBL9658504 0.83 TAS1R3 (0.53) PARP10ALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL11662636 0.83 PARP10 (0.38) CYP19A1PARP10POLBTDP1TSHR
SCHEMBL6836501 0.82 PARP10 (0.66) PARP10POLBKMT2AGLAALDH1A1
SCHEMBL4763620 0.81 LDHA (0.52) PARP10POLBTDP1TSHRKMT2A
SCHEMBL28492939 0.81 CYP1A2 (0.46) POLBTDP1TSHRKMT2AMAPK1
SCHEMBL316898 0.81 MTNR1A (0.50) KMT2AALDH1A1CYP3A4TP53CYP1A2
SCHEMBL3838993 0.80 ALDH1A1 (0.40) CYP19A1PARP10POLBTDP1TSHR
SCHEMBL2881391 0.80 TDP1 (0.52) PARP10POLBTDP1TSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105102456-B Azaquinazoline inhibitors of atypical protein kinase C 癌症研究技术有限公司 2017-11-14 CN disclosed
CN-105102456-A Azaquinazoline inhibitors of atypical protein kinase C IGNYTA INC 2015-11-25 CN disclosed