SCHEMBL28045892

SCHEMBL28045892

O=C1Nc2ccc(C(c3ccccc3)c3ccccc3)cc2C1=O

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAOA P21397 9/20 0.58
MAOB P27338 9/20 0.58
TGM2 P21980 5/20 0.50
CES1 P23141 3/20 0.50
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA9 Q16790 1/20 0.46
ALDH1A1 P00352 1/20 0.46
CASP3 P42574 2/20 0.45
CAPN9 O14815 1/20 0.45
SLC6A11 P48066 1/20 0.44
CASP2 P42575 1/20 0.44
CASP7 P55210 1/20 0.44
CASP6 P55212 1/20 0.44
CASP8 Q14790 1/20 0.44
PDE3B Q13370 1/20 0.44
PDE3A Q14432 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4444879 0.77 TGM2 (0.55) MAOAMAOBTGM2CES1CA12
SCHEMBL11081844 0.74 MAOA (0.47) MAOAMAOBTGM2CES1CA12
SCHEMBL2789935 0.74 MAOA (1.00) MAOAMAOBTGM2CES1CA12
SCHEMBL5330038 0.73 TGM2 (0.53) MAOAMAOBTGM2CES1CA12
SCHEMBL16111115 0.72 CES1 (0.53) MAOAMAOBTGM2CES1CA12
Isatin SCHEMBL28365971 0.72 MAOA (0.95) MAOAMAOBTGM2CES1ALDH1A1
SCHEMBL1767901 0.71 TGM2 (0.50) MAOAMAOBTGM2CES1CA12
SCHEMBL4967546 0.71 ALDH1A1 (0.55) MAOAMAOBTGM2CES1CA12
SCHEMBL9330149 0.70 MAOA (0.58) MAOAMAOBTGM2CES1CA12
Isatin SCHEMBL34016 0.69 MAOA (1.00) MAOAMAOBTGM2CES1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102256983-B Spirooxindole compounds and their use as therapeutic agents 泽农医药公司 2017-04-05 CN disclosed
CN-105218565-A Spiral shell oxindole compounds and the purposes as therapeutical agent thereof XENON PHARMACEUTICALS INC 2016-01-06 CN disclosed
CN-105175433-A Spiro-oxindole compounds and their use as therapeutic agents XENON PHARMACEUTICALS INC 2015-12-23 CN disclosed