SCHEMBL28046609

SCHEMBL28046609

NC(=O)c1cc2ccc(-c3ccc(Br)cc3)nc2[nH]1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.43
RXFP1 Q9HBX9 2/20 0.41
CDC7 O00311 1/20 0.39
MCL1 Q07820 3/20 0.39
MAP2K1 Q02750 1/20 0.39
LMNA P02545 1/20 0.39
ROCK2 O75116 2/20 0.39
ROCK1 Q13464 2/20 0.39
ACR P10323 1/20 0.39
CHEK2 O96017 1/20 0.38
GRM2 Q14416 1/20 0.37
EPRS1 P07814 1/20 0.36
NUDT1 P36639 1/20 0.36
SNCA P37840 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28046616 0.86 PARP1 (0.47) CDC7ROCK2ROCK1ACRCHEK2
SCHEMBL28046664 0.86 MAP4K4 (0.46) CASP1CHEK2NUDT1
SCHEMBL28046684 0.83 KMO (0.44) CASP1ROCK2ROCK1NUDT1
SCHEMBL28046610 0.82 ROCK2 (0.54) CASP1LMNAROCK2ROCK1
SCHEMBL28046613 0.81 CDK5 (0.41) ROCK2ROCK1CHEK2
SCHEMBL28046667 0.81 KMO (0.42) CHEK2NUDT1
SCHEMBL28046677 0.81 ALPL (0.45) ROCK2ROCK1CHEK2
SCHEMBL28046611 0.79 MAPT (0.54) RXFP1MCL1ROCK2ROCK1
SCHEMBL30988404 0.78 ROCK2 (0.58) ROCK2ROCK1
SCHEMBL28046612 0.77 DHODH (0.46) CDC7ROCK2ROCK1NUDT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105294688-A 6-chlorine-N-(substituted benzyl)-1H-pyrrolo[2,3-b]pyridine-2-amide compound and preparation method as well as application thereof UNIV BEIJING TECHNOLOGY 2016-02-03 CN disclosed