SCHEMBL28046684

SCHEMBL28046684

NC(=O)c1cc2ccc(-c3ccc(F)c(F)c3)nc2[nH]1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 2/20 0.44
IDO1 P14902 1/20 0.44
HSD17B14 Q9BPX1 3/20 0.38
NUDT1 P36639 1/20 0.38
TRPV3 Q8NET8 1/20 0.38
JAK2 O60674 1/20 0.36
ROCK2 O75116 3/20 0.36
ROCK1 Q13464 3/20 0.36
CASP1 P29466 1/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
PSMD14 O00487 1/20 0.36
MAPT P10636 2/20 0.35
CYP1A2 P05177 2/20 0.35
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C8 P10632 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28046616 0.86 PARP1 (0.47) HSD17B14ROCK2ROCK1ALDH1A1RAB9A
SCHEMBL28046609 0.83 CASP1 (0.43) NUDT1ROCK2ROCK1CASP1
SCHEMBL28046664 0.83 MAP4K4 (0.46) KMONUDT1CASP1MAPTRAB9A
SCHEMBL28046665 0.83 HPGDS (0.51) KMOIDO1NUDT1ROCK2ROCK1
SCHEMBL28046667 0.81 KMO (0.42) KMONUDT1MEN1KMT2AMAPT
SCHEMBL28046677 0.81 ALPL (0.45) HSD17B14ROCK2ROCK1MAPTALDH1A1
SCHEMBL28046611 0.79 MAPT (0.54) ROCK2ROCK1MEN1KMT2AMAPT
SCHEMBL28046615 0.78 PARP1 (0.49) NUDT1RAB9A
SCHEMBL28046610 0.77 ROCK2 (0.54) JAK2ROCK2ROCK1CASP1MEN1
SCHEMBL28046612 0.77 DHODH (0.46) KMONUDT1ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105294688-A 6-chlorine-N-(substituted benzyl)-1H-pyrrolo[2,3-b]pyridine-2-amide compound and preparation method as well as application thereof UNIV BEIJING TECHNOLOGY 2016-02-03 CN disclosed