SCHEMBL28046677

SCHEMBL28046677

Cc1ccc(-c2ccc3cc(C(N)=O)[nH]c3n2)cc1C

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALPL P05186 2/20 0.45
CA9 Q16790 1/20 0.45
CHEK2 O96017 4/20 0.41
CCNC P24863 2/20 0.39
CDK8 P49336 2/20 0.39
ROCK2 O75116 7/20 0.38
ROCK1 Q13464 7/20 0.38
TP53 P04637 1/20 0.37
MAPT P10636 1/20 0.37
ALDH1A1 P00352 1/20 0.37
RIPK1 Q13546 1/20 0.36
HSD17B1 P14061 1/20 0.36
HSD17B2 P37059 1/20 0.36
HSD17B14 Q9BPX1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28046612 0.83 DHODH (0.46) ROCK2ROCK1
SCHEMBL28046611 0.82 MAPT (0.54) ROCK2ROCK1MAPTALDH1A1
SCHEMBL28046667 0.81 KMO (0.42) CHEK2CCNCCDK8MAPT
SCHEMBL28046684 0.81 KMO (0.44) ROCK2ROCK1MAPTALDH1A1HSD17B14
SCHEMBL28046616 0.81 PARP1 (0.47) ALPLCHEK2ROCK2ROCK1ALDH1A1
SCHEMBL28046609 0.81 CASP1 (0.43) CHEK2ROCK2ROCK1
SCHEMBL28046664 0.81 MAP4K4 (0.46) ALPLCHEK2CCNCCDK8MAPT
SCHEMBL28046610 0.80 ROCK2 (0.54) ALPLCA9ROCK2ROCK1TP53
SCHEMBL28046662 0.80 JAK2 (0.43) CCNCCDK8ROCK2ROCK1MAPT
SCHEMBL28046613 0.79 CDK5 (0.41) CHEK2ROCK2ROCK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105294688-A 6-chlorine-N-(substituted benzyl)-1H-pyrrolo[2,3-b]pyridine-2-amide compound and preparation method as well as application thereof UNIV BEIJING TECHNOLOGY 2016-02-03 CN disclosed