SCHEMBL28050469

SCHEMBL28050469

C[C@@](O)(C(=O)Nc1ccccc1)C(F)(F)F

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 15/20 1.00
PDK2 Q15119 15/20 1.00
PDK3 Q15120 15/20 1.00
PDK4 Q16654 15/20 1.00
ABCC9 O60706 7/20 0.77
ABCC8 Q09428 7/20 0.77
KCNJ11 Q14654 7/20 0.77
KCNJ8 Q15842 7/20 0.77
ABCB11 O95342 1/20 0.77
MEN1 O00255 1/20 0.72
CYP1A2 P05177 1/20 0.72
CYP3A4 P08684 1/20 0.72
CYP2D6 P10635 1/20 0.72
TSHR P16473 1/20 0.72
CYP2C19 P33261 1/20 0.72
KMT2A Q03164 1/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6359557 1.00 PDK1 (1.00) PDK1PDK2PDK3PDK4ABCC9
Zd-6169 SCHEMBL2123811 0.87 ABCC9 (1.00) PDK1PDK2PDK3PDK4ABCC9
Zd-6169 SCHEMBL4261046 0.87 ABCC9 (1.00) PDK1PDK2PDK3PDK4ABCC9
SCHEMBL2128828 0.85 ABCC9 (1.00) PDK1PDK2PDK3PDK4ABCC9
SCHEMBL5317709 0.84 PDK1 (0.75) PDK1PDK2PDK3PDK4ABCC9
SCHEMBL8489691 0.84 ABCC9 (0.74) PDK1PDK2PDK3PDK4ABCC9
SCHEMBL9709058 0.83 PDK1 (0.71) PDK1PDK2PDK3PDK4ABCC9
SCHEMBL16212234 0.82 PDK1 (0.70) PDK1PDK2PDK3PDK4ABCC9
SCHEMBL8867579 0.81 PDK1 (0.71) PDK1PDK2PDK3PDK4ABCC9
SCHEMBL3129785 0.80 PDK1 (0.67) PDK1PDK2PDK3PDK4ABCC9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103951584-B Derivative of 3-chloro-N-phenyl-4-(the fluoro-2-methyl of 3,3,3-tri--2-hydroxypropanamide base) benzamide and preparation method thereof and application TSINGHUA UNIVERSITY (CN) 2016-02-10 CN disclosed