SCHEMBL28053364

SCHEMBL28053364

Cc1ccc2c(c1)C(=O)C(=O)N2Cc1ccc(Br)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 1.00
HSP90AA1 P07900 1/20 0.70
TP53 P04637 4/20 0.67
MAPT P10636 3/20 0.67
ALDH1A1 P00352 6/20 0.66
ALDH3A1 P30838 6/20 0.66
ALDH2 P05091 4/20 0.66
CHRM5 P08912 2/20 0.65
CHRM1 P11229 1/20 0.65
CHRM3 P20309 1/20 0.65
PARK7 Q99497 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16329852 0.91 ACHE (0.83) ACHEHSP90AA1TP53MAPTALDH1A1
SCHEMBL28053294 0.88 ACHE (1.00) ACHEALDH1A1ALDH3A1ALDH2CHRM5
SCHEMBL4597228 0.87 ACHE (0.77) ACHEHSP90AA1TP53MAPTALDH1A1
SCHEMBL22410741 0.86 ACHE (0.75) ACHEHSP90AA1TP53MAPTALDH1A1
SCHEMBL14047967 0.86 ACHE (0.75) ACHEHSP90AA1TP53MAPTALDH1A1
SCHEMBL578250 0.85 ACHE (0.74) ACHEHSP90AA1TP53MAPTALDH1A1
SCHEMBL28053291 0.85 ACHE (0.74) ACHEHSP90AA1TP53MAPTALDH1A1
SCHEMBL4597560 0.81 ACHE (0.86) ACHEALDH1A1ALDH3A1ALDH2CHRM5
SCHEMBL5659265 0.79 ALDH1A1 (1.00) ACHEALDH1A1ALDH3A1ALDH2CHRM5
SCHEMBL2056299 0.79 CHRM5 (0.81) ACHEHSP90AA1TP53MAPTCHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105237521-B A kind of cumarin-isatin type compound and its preparation method and purposes 诸暨市志缇生物科技有限公司 2018-08-24 CN disclosed
CN-105541808-A Metronidazole-isatin type compound as well as preparation method and application thereof UNIV JISHOU 2016-05-04 CN disclosed
CN-105237521-A Coumarin-isatin type compounds, and preparation method and purpose thereof UNIV JISHOU 2016-01-13 CN disclosed