SCHEMBL28056270

SCHEMBL28056270

Nc1ccc(OC(F)(F)F)c(Cl)c1O

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.33
SLC1A5 Q15758 2/20 0.33
EPHX2 P34913 1/20 0.33
ACLY P53396 1/20 0.32
KMO O15229 2/20 0.31
AKR1C2 P52895 1/20 0.31
AKR1C1 Q04828 1/20 0.31
GRIN2B Q13224 1/20 0.31
NOS3 P29474 1/20 0.30
NOS1 P29475 1/20 0.30
NOS2 P35228 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8074941 0.82 PDE2A (0.33) PDE2ASLC1A5EPHX2KMOGRIN2B
SCHEMBL30127239 0.79 MPL (0.36) PDE2ASLC1A5EPHX2
SCHEMBL19485985 0.78 ALDH1A1 (0.35) PDE2ASLC1A5
SCHEMBL16798567 0.78 PDE2A (0.30) PDE2ASLC1A5
SCHEMBL10710521 0.77 EPHX2 (0.37) PDE2ASLC1A5EPHX2KMOGRIN2B
SCHEMBL28056190 0.75 IDO1 (0.44)
SCHEMBL28056275 0.74 GRIN2B (0.36) PDE2ASLC1A5EPHX2ACLYKMO
SCHEMBL28056195 0.73 MPL (0.40) GRIN2B
SCHEMBL7937713 0.73 MPL (0.40) GRIN2B
SCHEMBL5328165 0.72 KMO (0.34) EPHX2KMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105431427-B Novel PDE 4 inhibitor 明治制果药业株式会社 2017-12-08 CN disclosed
CN-105431427-A Novel PDE4 inhibitor MEIJI SEIKA PHARMA CO LTD 2016-03-23 CN disclosed