SCHEMBL28061520

SCHEMBL28061520

C[CH]c1cc(C)c(Sc2ccc(OC)cc2)c(C)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TUBB1 Q9H4B7 2/20 0.45
PTGS2 P35354 3/20 0.42
PTGS1 P23219 2/20 0.42
ALOX5 P09917 2/20 0.42
CYP1A1 P04798 2/20 0.42
CYP1A2 P05177 2/20 0.42
CYP1B1 Q16678 2/20 0.42
AR P10275 2/20 0.39
PTGIR P43119 1/20 0.39
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 2/20 0.39
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
CYP3A4 P08684 1/20 0.39
TSHR P16473 1/20 0.39
RELA Q04206 1/20 0.38
HAO1 Q9UJM8 1/20 0.37
AKR1B1 P15121 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.37
ESR1 P03372 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18723690 0.79 TDP1 (0.47) PTGS2PTGS1ARPTGIRALDH1A1
SCHEMBL28061534 0.75 PTGIR (0.41) PTGS2PTGS1ARPTGIRALDH1A1
SCHEMBL18723868 0.75 PTGS1 (0.39) PTGS2PTGS1CYP1A1CYP1A2CYP1B1
SCHEMBL18723828 0.74 PTGS1 (0.41) PTGS2PTGS1ARPTGIRALDH1A1
SCHEMBL27916620 0.74 PTGS1 (0.39) TUBB1PTGS2PTGS1CYP1A1CYP1A2
SCHEMBL27916545 0.74 TUBB1 (0.49) TUBB1PTGS2PTGS1ALOX5CYP1A1
SCHEMBL28061531 0.73 PTGS1 (0.38) TUBB1PTGS2PTGS1CYP1A1CYP1A2
SCHEMBL28061523 0.71 ALDH1A1 (0.46) PTGS2PTGS1PTGIRALDH1A1KDM4E
SCHEMBL482369 0.71 CA1 (0.65) CYP1A1CYP1A2CYP1B1PTGIRALDH1A1
SCHEMBL28061510 0.70 F2RL1 (0.51) PTGS2PTGS1ALOX5CYP1A2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105906617-B Modulators of HEC1 activity and methods thereof 泰纬生命科技股份有限公司 2018-09-04 CN disclosed
CN-105906617-A Modulators of HEC1 activity and methods thereof 泰纬生命科技股份有限公司 2016-08-31 CN disclosed
CN-103038231-B Modulators of HEC1 activity and methods thereof Taivex Therapeutics Corp. (CN) 2016-04-20 CN disclosed