SCHEMBL28061510

SCHEMBL28061510

COc1ccc(Sc2c(C)cc(CCC(=O)CCc3cc(C)c(Sc4ccc(OC)cc4)c(C)c3)cc2C)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2RL1 P55085 1/20 0.51
AKR1B1 P15121 1/20 0.43
PTGDR2 Q9Y5Y4 1/20 0.43
NFKB1 P19838 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43
SLC5A1 P13866 1/20 0.42
SLC5A2 P31639 1/20 0.42
ALOX5 P09917 1/20 0.42
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
MAPT P10636 3/20 0.40
KDM4E B2RXH2 1/20 0.40
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
MAOA P21397 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A3 Q01959 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28061531 0.81 PTGS1 (0.38) AKR1B1PTGDR2MAPTKDM4ECYP1A2
SCHEMBL27986391 0.78 F2RL1 (0.55) F2RL1NFKB1NFKB2RELASLC5A1
SCHEMBL28061534 0.78 PTGIR (0.41) AKR1B1PTGDR2NPC1RAB9AMAPT
SCHEMBL28061523 0.76 ALDH1A1 (0.46) AKR1B1PTGDR2RAB9AMAPTKDM4E
SCHEMBL7329940 0.75 F2RL1 (0.85) F2RL1NFKB1NFKB2RELASLC5A1
SCHEMBL28154615 0.74 RAPGEF4 (0.67) F2RL1MAPTTP53CYP3A4SMN1; SMN2
SCHEMBL28061511 0.73 F2RL1 (0.49) F2RL1NFKB1NFKB2RELASLC5A1
SCHEMBL18723690 0.72 TDP1 (0.47) AKR1B1PTGDR2MAPTKDM4ECYP3A4
SCHEMBL28833020 0.72 AKR1B1 (0.43) AKR1B1PTGDR2MAPTALDH1A1POLB
SCHEMBL7328673 0.71 F2RL1 (0.56) F2RL1AKR1B1NFKB1NFKB2RELA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105906617-A Modulators of HEC1 activity and methods thereof 泰纬生命科技股份有限公司 2016-08-31 CN disclosed
CN-103038231-B Modulators of HEC1 activity and methods thereof Taivex Therapeutics Corp. (CN) 2016-04-20 CN disclosed