SCHEMBL28072002

SCHEMBL28072002

C=Cc1ccc(N2CC[CH]CC2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.46
TRIM24 O15164 1/20 0.44
TRIM33 Q9UPN9 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.42
KDM4E B2RXH2 3/20 0.42
FURIN P09958 1/20 0.41
HTR1A P08908 1/20 0.39
HTR2A P28223 1/20 0.39
PTGS2 P35354 3/20 0.38
MAPT P10636 6/20 0.38
KMT2A Q03164 2/20 0.37
ACHE P22303 1/20 0.37
MEN1 O00255 1/20 0.37
TDP1 Q9NUW8 2/20 0.36
TSHR P16473 1/20 0.36
GFER P55789 2/20 0.35
LMNA P02545 1/20 0.35
MAPK1 P28482 1/20 0.35
HTT P42858 1/20 0.35
F2 P00734 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL628551 0.89 ALDH1A1 (0.58) ALDH1A1TRIM24TRIM33SMN1; SMN2KDM4E
SCHEMBL98716 0.83 TRIM24 (0.63) ALDH1A1TRIM24TRIM33SMN1; SMN2KDM4E
SCHEMBL817331 0.81 ALDH1A1 (0.64) ALDH1A1TRIM24TRIM33SMN1; SMN2KDM4E
SCHEMBL609198 0.81 ALDH1A1 (0.64) ALDH1A1TRIM24TRIM33SMN1; SMN2KDM4E
SCHEMBL99032 0.79 ALDH1A1 (0.69) ALDH1A1SMN1; SMN2KDM4EMAPTKMT2A
SCHEMBL2904812 0.79 ALDH1A1 (0.54) ALDH1A1SMN1; SMN2KDM4EMAPTKMT2A
SCHEMBL13920008 0.79 KDM4E (0.54) ALDH1A1TRIM24TRIM33SMN1; SMN2KDM4E
SCHEMBL14394962 0.78 ADRB1 (0.57) ALDH1A1KDM4ETSHRLMNA
SCHEMBL21411223 0.75 GAA (0.62) ALDH1A1SMN1; SMN2KDM4EHTR1AHTR2A
SCHEMBL17923046 0.73 ME2 (0.47) ALDH1A1TRIM24TRIM33SMN1; SMN2PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105722823-A NOVEL CYTOCHROME P450 INHIBITORS AND THEIR METHOD OF USE 科尔泰多公众股份公司 2016-06-29 CN disclosed