SCHEMBL28073294

SCHEMBL28073294

Cc1cc(C)cc(Cc2ncc([N+](=O)[O-])c(N)n2)c1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
RAB9A P51151 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.37
PIN1 Q13526 2/20 0.36
TSHR P16473 3/20 0.36
CYP3A4 P08684 1/20 0.36
RECQL P46063 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
GPR35 Q9HC97 1/20 0.36
PRKCQ Q04759 1/20 0.34
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28802640 0.77 ALDH1A1 (0.46) ALDH1A1RAB9ASMN1; SMN2PRKCQ
SCHEMBL28081097 0.76 TSHR (0.44) ALDH1A1LMNAMAPTTDP1SMN1; SMN2
SCHEMBL14641049 0.76 PIN1 (0.40) ALDH1A1LMNAMAPTHTTRAB9A
SCHEMBL2632674 0.72 ALDH1A1 (0.41) ALDH1A1LMNAMAPTHTTRAB9A
SCHEMBL27088207 0.70 USP1 (0.40)
SCHEMBL5789457 0.68 HASPIN (0.44) ALDH1A1LMNAMAPTHTTRAB9A
SCHEMBL2950586 0.68 LMNA (0.42) ALDH1A1LMNAMAPTHTTRAB9A
SCHEMBL1414668 0.68 DHFR (0.53) ALDH1A1LMNAMAPTHTTRAB9A
SCHEMBL27258254 0.67 TDP1 (0.42) ALDH1A1LMNAMAPTHTTRAB9A
SCHEMBL1194395 0.65 PIN1 (0.52) PIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105814056-B purine derivatives as modulators of TNF activity UCB生物制药私人有限公司 2017-10-10 CN disclosed
CN-105814056-A Purine derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed