SCHEMBL28077287

SCHEMBL28077287

CN1CCC[C@H]1CCC1NCCc2ccc(-c3cc(N)ccc3S(N)(=O)=O)cc21

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 8/20 0.36
TBXA2R P21731 1/20 0.34
CHRNB2 P17787 1/20 0.32
CHRNA4 P43681 1/20 0.32
HTR7 P34969 1/20 0.32
METAP2 P50579 4/20 0.32
KCNH2 Q12809 2/20 0.31
HTR6 P50406 1/20 0.31
NOS3 P29474 2/20 0.31
NOS1 P29475 2/20 0.31
NOS2 P35228 2/20 0.31
CHRNB4 P30926 1/20 0.31
CHRNA3 P32297 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2402408 0.81 HTR7 (0.40) HTR7
SCHEMBL2405712 0.81 HTR7 (0.40) HTR7
SCHEMBL28077422 0.81 CHRM3 (0.33) CHRM3METAP2
Hydrochloric Acid SCHEMBL14686044 0.81 HTR7 (0.39) HTR7NOS3NOS1NOS2
SCHEMBL28077284 0.65 PNMT (0.55)
SCHEMBL14208854 0.65 KCNH2 (0.44) CHRM3CHRNB2CHRNA4HTR7KCNH2
SCHEMBL28001951 0.65 HRH3 (0.40) CHRM3HTR7METAP2
SCHEMBL2675396 0.64 KCNH2 (0.57) CHRM3CHRNB2CHRNA4HTR7KCNH2
SCHEMBL2493535 0.64 PDE5A (0.38) HTR7METAP2HTR6
SCHEMBL2675587 0.64 NOS3 (0.57) CHRM3CHRNB2CHRNA4HTR7KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105764510-A An H3 receptor antagonist combined with a cholinesterase inhibitor for use in the treatment of alzheimer's disease 赛诺菲 2016-07-13 CN disclosed