SCHEMBL28077415

SCHEMBL28077415

Cc1ccccc1-c1nc(O)c(O)s1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPM8 Q7Z2W7 2/20 0.50
ALDH1A1 P00352 3/20 0.41
HTR2B P41595 1/20 0.41
NPC1 O15118 4/20 0.39
RAB9A P51151 3/20 0.39
LMNA P02545 2/20 0.39
ALOX5 P09917 1/20 0.39
HPGD P15428 3/20 0.39
MAPT P10636 3/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 1/20 0.39
GAA P10253 1/20 0.39
STAT6 P42226 1/20 0.39
HIF1A Q16665 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
SMN1; SMN2 Q16637 3/20 0.38
NFKB1 P19838 2/20 0.38
NFKB2 Q00653 2/20 0.38
RELA Q04206 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28077207 0.79 ALDH1A1 (0.46) ALDH1A1NPC1RAB9AALOX5MAPT
SCHEMBL13801072 0.76 ALDH1A1 (0.42) TRPM8ALDH1A1NPC1RAB9ALMNA
SCHEMBL28077336 0.76 HDAC9 (0.39) TRPM8LMNAALOX5MAPT
SCHEMBL17374828 0.75 TRPM8 (0.55) TRPM8ALDH1A1MAPTKDM4E
SCHEMBL4297511 0.73 HTR2B (0.42) TRPM8ALDH1A1HTR2BNPC1RAB9A
SCHEMBL8989405 0.73 TRPM8 (0.36) TRPM8ALDH1A1HTR2BNPC1RAB9A
SCHEMBL1954805 0.72 ALOX5 (0.56) TRPM8ALDH1A1ALOX5MEN1KMT2A
SCHEMBL28077372 0.71 SLC9A1 (0.35) TRPM8ALDH1A1NPC1RAB9ALMNA
SCHEMBL17374836 0.71 TRPM8 (0.79) TRPM8ALDH1A1NPC1RAB9ALMNA
SCHEMBL23176718 0.70 ALDH1A1 (0.39) TRPM8ALDH1A1NPC1RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104334544-B Benzimidazole proline derivative 埃科特莱茵药品有限公司 2016-10-19 CN disclosed