SCHEMBL28111098

SCHEMBL28111098

CC(=O)ONc1cc(C(O)CCC2CC2)ccc1F

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACACB O00763 5/20 0.36
KLKB1 P03952 11/20 0.34
CCR5 P51681 1/20 0.34
ADRB1 P08588 1/20 0.33
ADRA2A P08913 1/20 0.33
ADRB3 P13945 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28111673 0.87 ACACB (0.35) ACACBKLKB1
SCHEMBL28111162 0.87 ACACB (0.37) ACACBKLKB1
SCHEMBL17064969 0.83 KLKB1 (0.39) KLKB1
SCHEMBL17064972 0.81 GLA (0.41) KLKB1CCR5
SCHEMBL23429072 0.79 ADRB1 (0.35) KLKB1ADRB1ADRA2AADRB3ADRA2B
SCHEMBL28534568 0.74 ALDH1A1 (0.39) CCR5ADRB1ADRA2AADRB3ADRA2B
SCHEMBL25668311 0.74 ADRB1 (0.38) CCR5ADRB1ADRA2AADRB3ADRA2B
SCHEMBL22394359 0.72 ADRB1 (0.35) CCR5ADRB1ADRA2AADRB3ADRA2B
SCHEMBL17064475 0.72 ADRB1 (0.35) CCR5ADRB1ADRA2AADRB3ADRA2B
SCHEMBL28938019 0.71 KLKB1 (0.54) KLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106257976-A Human plasma kallikrein inhibitors 拜奥克里斯特制药公司 2016-12-28 CN disclosed