SCHEMBL28116044

SCHEMBL28116044

CCOC(=O)C(C=CCl)C(C)=O

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.39
LMNA P02545 1/20 0.39
HSD17B10 Q99714 1/20 0.39
GLO1 Q04760 1/20 0.35
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
ALOX15 P16050 1/20 0.33
MGAM O43451 1/20 0.33
GAA P10253 1/20 0.33
SI P14410 1/20 0.33
MGAM2 Q2M2H8 1/20 0.33
SOAT1 P35610 1/20 0.33
HCAR2 Q8TDS4 1/20 0.32
NPSR1 Q6W5P4 1/20 0.31
TRPA1 O75762 1/20 0.31
HPGD P15428 1/20 0.30
PIN1 Q13526 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6070239 0.77 ALDH1A1 (0.44) ALDH1A1LMNAHSD17B10GLO1CYP2D6
SCHEMBL9620433 0.76 GLO1 (0.36) ALDH1A1LMNAHSD17B10GLO1CYP2D6
SCHEMBL9620431 0.76 GLO1 (0.36) ALDH1A1LMNAHSD17B10GLO1CYP2D6
SCHEMBL15046951 0.75 ALDH1A1 (0.42) ALDH1A1LMNAHSD17B10GLO1CYP2D6
SCHEMBL18431955 0.74 FBP1 (0.36) ALDH1A1LMNAHSD17B10GLO1CYP2C9
SCHEMBL28244012 0.73 CYP2D6 (0.36) ALDH1A1LMNAHSD17B10GLO1CYP2D6
SCHEMBL11461030 0.72 ALDH1A1 (0.39) ALDH1A1LMNAHSD17B10GLO1CYP2D6
SCHEMBL10467804 0.72 ALDH1A1 (0.39) ALDH1A1LMNAHSD17B10GLO1CYP2D6
SCHEMBL2915798 0.70 ALDH1A1 (0.42) ALDH1A1LMNAHSD17B10GLO1CYP2D6
SCHEMBL10275655 0.69 ALDH1A1 (0.46) ALDH1A1LMNAHSD17B10GLO1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109354584-A The method of one pot process 2- (4- hydroxy phenyl) -4- methyl-1,3-thiazole-5-carboxylic acid ethyl ester 湖北理工学院 2019-02-19 CN claimed
CN-108570017-A The synthesis of 2- amino-4-methylthiazole-5-carboxylates 西安格瑞德化工新材料有限公司 2018-09-25 CN claimed
CN-108218702-A The preparation method of 2- acetyl fluoride ethyl acetate 湖北卓熙氟化股份有限公司 2018-06-29 CN claimed
CN-105753858-B Heterocyclic compound and p27Kip1Decomposing inhibitor ASKA制药株式会社 2019-04-30 CN disclosed
CN-109574952-A A kind of synthetic method of febuxostat intermediate 安徽省庆云医药股份有限公司 2019-04-05 CN disclosed
CN-109574951-A A kind of preparation method of Febuxostat 安徽省庆云医药股份有限公司 2019-04-05 CN disclosed
CN-109575018-A A kind of anti-infective compounds 韩国巴斯德研究所 2019-04-05 CN disclosed
CN-105622637-B Thiazole simultaneously [3,2-b] -1,2,4- triazine -2- carboxylic acid derivates and its preparation method and application 沈阳药科大学 2018-09-25 CN disclosed
CN-108218702-A The preparation method of 2- acetyl fluoride ethyl acetate 湖北卓熙氟化股份有限公司 2018-06-29 CN disclosed
CN-105777664-B Carboxylate of 2 (2 benzyl hydrazono-) thiazole 5 and preparation method thereof and medical usage 湖南大学 2017-12-29 CN disclosed
CN-206570248-U A kind of continuous synthesis system of 4 chloroacetyl acetacetic ester 江苏诚信药业有限公司 2017-10-20 CN disclosed
CN-104781258-B Hydroxy-substituted imidazo [1,2-a ] pyridinecarboxamides and their use as soluble guanylate cyclase stimulators 拜耳制药股份公司 2017-09-22 CN disclosed
CN-105745212-B Spiro derivatives of substituted 4, 5-dihydropyrazolo [3,4-c ] pyridin-2-ones and uses thereof 四川海思科制药有限公司 2017-09-12 CN disclosed
CN-106748764-A The continuous synthesis system and method for a kind of 4 chloroacetyl acetacetic ester 江苏诚信药业有限公司 2017-05-31 CN disclosed
CN-106752470-A A kind of skin coating 安徽钰锦生态木材料有限公司 2017-05-31 CN disclosed
CN-105026392-B 4,5-dihydro-pyrazolo [3, 4-c] pyrid-2-ones, preparation method and application thereof 四川海思科制药有限公司 2017-05-10 CN disclosed
CN-104529935-B Method for synthesizing ethyl 2-(3-aldehyde-4-isobutyloxyphenyl)-4-methylthiazole-5-formate 浙江华义医药有限公司 2017-04-12 CN disclosed
CN-106543139-A A kind of triadimefon compound and application thereof 沈阳中化农药化工研发有限公司 2017-03-29 CN disclosed
CN-106459037-A Enantiomers of the n-(2-amino-5-fluoro-2-methylpentyl)-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridine-3-carboxamide, as well as of the di- and trifluoro derivatives for the treatment of cardiovascular diseases 拜耳医药股份有限公司 2017-02-22 CN disclosed
CN-106414440-A Aryl and heteroaryl substituted imidazo [1,2-a ] pyridine-3-carboxamides and their use 拜耳制药股份公司 2017-02-15 CN disclosed